TN2013000179A1 - Piperidinone carboxamide azaindane cgrp receptor antagonists - Google Patents

Piperidinone carboxamide azaindane cgrp receptor antagonists

Info

Publication number: TN2013000179A1
Authority: TN; Tunisia
Prior art keywords: receptor antagonists; cgrp receptor; piperidinone carboxamide; carboxamide azaindane; piperidinone
Prior art date: 2011-11-10

Application number

TNP2013000179A

Other languages

English (en)

Inventor

Ian M Bell

Mark E Fraley

Steven N Gallicchio

Anthony Ginnetti

Helen J Mitchell

Daniel V Paone

Donnette D Staas

Cheng Wang

C Blair Zartman

Heather E Stevenson

Original Assignee

Merck Sharp & Dohme

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2011-11-10

Filing date

2013-04-24

Publication date

2014-11-10

2011-11-10 Priority claimed from PCT/US2011/060081 external-priority patent/WO2012064910A1/fr

2013-04-24 Application filed by Merck Sharp & Dohme filed Critical Merck Sharp & Dohme

2014-11-10 Publication of TN2013000179A1 publication Critical patent/TN2013000179A1/fr

Links

108010078311 Calcitonin Gene-Related Peptide Receptors Proteins 0.000 title abstract 2
102000008323 calcitonin gene-related peptide receptor activity proteins Human genes 0.000 title 1
150000003857 carboxamides Chemical class 0.000 title 1
LPAGFVYQRIESJQ-UHFFFAOYSA-N indoline Chemical compound C1=CC=C2NCCC2=C1 LPAGFVYQRIESJQ-UHFFFAOYSA-N 0.000 title 1
XUWHAWMETYGRKB-UHFFFAOYSA-N piperidin-2-one Chemical compound O=C1CCCCN1 XUWHAWMETYGRKB-UHFFFAOYSA-N 0.000 title 1
239000002464 receptor antagonist Substances 0.000 title 1
229940044551 receptor antagonist Drugs 0.000 title 1
108090000932 Calcitonin Gene-Related Peptide Proteins 0.000 abstract 2
102100025588 Calcitonin gene-related peptide 1 Human genes 0.000 abstract 2
150000001875 compounds Chemical class 0.000 abstract 2
102000014468 Calcitonin Gene-Related Peptide Receptors Human genes 0.000 abstract 1
208000019695 Migraine disease Diseases 0.000 abstract 1
239000005557 antagonist Substances 0.000 abstract 1
201000010099 disease Diseases 0.000 abstract 1
230000006806 disease prevention Effects 0.000 abstract 1
208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
206010027599 migraine Diseases 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
239000008194 pharmaceutical composition Substances 0.000 abstract 1
-1 piperidinone carboxamide azaindane derivatives Chemical class 0.000 abstract 1
230000002265 prevention Effects 0.000 abstract 1

Landscapes

Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

TNP2013000179A 2011-11-10 2013-04-24 Piperidinone carboxamide azaindane cgrp receptor antagonists TN2013000179A1 (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
PCT/US2011/060081 WO2012064910A1 (fr)	2010-11-12	2011-11-10	Antagonistes du récepteur cgrp de pipéridinone carboxamide azaindane

Publications (1)

Publication Number	Publication Date
TN2013000179A1 true TN2013000179A1 (en)	2014-11-10

Family

ID=54360614

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
TNP2013000179A TN2013000179A1 (en)	2011-11-10	2013-04-24	Piperidinone carboxamide azaindane cgrp receptor antagonists

Country Status (1)

Country	Link
TN (1)	TN2013000179A1 (fr)

2013
- 2013-04-24 TN TNP2013000179A patent/TN2013000179A1/fr unknown

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