NO20063636L - Muskariniske acetylkolinrecptoorantagonister - Google Patents
Muskariniske acetylkolinrecptoorantagonisterInfo
- Publication number
- NO20063636L NO20063636L NO20063636A NO20063636A NO20063636L NO 20063636 L NO20063636 L NO 20063636L NO 20063636 A NO20063636 A NO 20063636A NO 20063636 A NO20063636 A NO 20063636A NO 20063636 L NO20063636 L NO 20063636L
- Authority
- NO
- Norway
- Prior art keywords
- acetylcholine receptor
- receptor antagonists
- muscarinic acetylcholine
- muscarinic
- methods
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
- C07D451/06—Oxygen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US53609204P | 2004-01-13 | 2004-01-13 | |
PCT/US2005/001333 WO2005067537A2 (fr) | 2004-01-13 | 2005-01-13 | Antagonistes des recepteurs muscariniques de l'acetylcholine |
Publications (1)
Publication Number | Publication Date |
---|---|
NO20063636L true NO20063636L (no) | 2006-10-04 |
Family
ID=34794385
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20063636A NO20063636L (no) | 2004-01-13 | 2006-08-11 | Muskariniske acetylkolinrecptoorantagonister |
Country Status (16)
Country | Link |
---|---|
US (1) | US20080249127A1 (fr) |
EP (1) | EP1711183A4 (fr) |
JP (1) | JP2007518740A (fr) |
KR (1) | KR20060129017A (fr) |
CN (1) | CN1929844A (fr) |
AR (1) | AR049464A1 (fr) |
AU (1) | AU2005204935A1 (fr) |
BR (1) | BRPI0506777A (fr) |
CA (1) | CA2552880A1 (fr) |
IL (1) | IL176775A0 (fr) |
MA (1) | MA28363A1 (fr) |
NO (1) | NO20063636L (fr) |
PE (1) | PE20050898A1 (fr) |
RU (1) | RU2006129289A (fr) |
TW (1) | TW200534855A (fr) |
WO (1) | WO2005067537A2 (fr) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2005087236A1 (fr) * | 2004-03-11 | 2005-09-22 | Glaxo Group Limited | Nouveaux antagonistes du recepteur de l'acetylcholine muscarinique m3 |
PE20060259A1 (es) | 2004-04-27 | 2006-03-25 | Glaxo Group Ltd | Compuestos de quinuclidina como antagonistas del receptor de acetilcolina muscarinico |
JP2007537261A (ja) * | 2004-05-13 | 2007-12-20 | グラクソ グループ リミテッド | ムスカリン性アセチルコリン受容体アンタゴニスト |
EP1765339A4 (fr) * | 2004-06-30 | 2009-09-02 | Glaxo Group Ltd | Antagonistes du recepteur muscarinique d'acetylcholine |
JP2008520579A (ja) * | 2004-11-15 | 2008-06-19 | グラクソ グループ リミテッド | 新規m3ムスカリン性アセチルコリン受容体アンタゴニスト |
US7479562B2 (en) | 2005-03-10 | 2009-01-20 | Theravance, Inc. | Biphenyl compounds useful as muscarinic receptor antagonists |
WO2007007282A2 (fr) * | 2005-07-11 | 2007-01-18 | Ranbaxy Laboratories Limited | Antagonistes des recepteurs muscariniques |
UY31637A1 (es) | 2008-02-06 | 2009-08-03 | Farmacoforos duales-antagonistas muscarinicos de pde4 | |
TW200946526A (en) | 2008-02-06 | 2009-11-16 | Glaxo Group Ltd | Dual pharmacophores-PDE4-muscarinic antagonistics |
TW200946525A (en) | 2008-02-06 | 2009-11-16 | Glaxo Group Ltd | Dual pharmacophores-PDE4-muscarinic antagonistics |
WO2010094643A1 (fr) | 2009-02-17 | 2010-08-26 | Glaxo Group Limited | Dérivés de quinoline et applications associées dans la rhinite et l'urticaire |
MY155212A (en) | 2009-04-30 | 2015-09-30 | Teijin Pharma Ltd | Quaternary ammonium salt compounds |
WO2014023325A1 (fr) * | 2012-08-06 | 2014-02-13 | Fondazione Istituto Italiano Di Tecnologia | Inhibiteurs de faah et de cox multicibles et leurs utilisations thérapeutiques |
KR101538846B1 (ko) * | 2013-07-30 | 2015-07-22 | 동아에스티 주식회사 | 신규한 바이페닐 유도체 및 그의 제조방법 |
CA3034535C (fr) | 2016-08-26 | 2021-07-06 | Dong-A St Co., Ltd. | Nouveau sel de (r)- (1-methylpyrrolidin-3-yl) methyl (3'-chloro -4'-fluoro- [1,1'-biphenyl]-2-yl) carbamate et forme cristalline de celui-ci |
KR102239776B1 (ko) * | 2016-08-26 | 2021-04-13 | 동아에스티 주식회사 | (r)-(1-메틸피롤리딘-3-일)메틸(3'-클로로-4'-플루오로-[1,1'-비페닐]-2-일)카바메이트의 신규염 및 이의 결정형 |
EP3710483A4 (fr) | 2017-11-16 | 2021-10-20 | XL-protein GmbH | Protéines de fusion vegfr/pdgfr pasylées et leur utilisation en thérapie |
WO2019110521A1 (fr) | 2017-12-04 | 2019-06-13 | Friedrich-Alexander-Universität Erlangen-Nürnberg | Ligands des récepteurs muscariniques à substitution fluorophényle ayant une sélectivité pour m3 sur m2 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IT1140998B (it) * | 1980-06-18 | 1986-10-10 | Valeas Ind Chimica E Farmaceut | Sali di endo-8-metil-8-sin-alchil-8-azoniabiciclo aperta par. quadrata 3.2.1. chiusa par. quadrata-ottan-3-alchilcarbossilati, processo per la loro preparazione e composizioni terapeutiche che li contengono come principio attivo |
EP0747355A4 (fr) * | 1994-02-10 | 1997-04-09 | Yamanouchi Pharma Co Ltd | Nouveau derive du carbamate et composition correspondante |
CA2415468A1 (fr) * | 2000-07-11 | 2003-01-10 | Yoshio Ogino | Derives d'ester |
US7365167B2 (en) * | 2001-11-26 | 2008-04-29 | Cell Matrix, Inc. | Humanized collagen antibodies and related methods |
MXPA04010966A (es) * | 2002-05-07 | 2005-01-25 | Neurosearch As | Derivados novedosos de biarilo diazabiciclico. |
US7041674B2 (en) * | 2002-11-26 | 2006-05-09 | Boehringer Ingelhiem Pharma Gmbh & Co. Kg | Carbamic acid esters with anticholinergic activity |
DE10255040A1 (de) * | 2002-11-26 | 2004-06-03 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Neue Carbaminsäureester mit anticholinerger Wirksamkeit |
US7232841B2 (en) * | 2003-04-07 | 2007-06-19 | Glaxo Group Limited | M3 muscarinic acetylcholine receptor antagonists |
-
2005
- 2005-01-11 TW TW094100746A patent/TW200534855A/zh unknown
- 2005-01-13 AR ARP050100118A patent/AR049464A1/es not_active Application Discontinuation
- 2005-01-13 PE PE2005000059A patent/PE20050898A1/es not_active Application Discontinuation
- 2005-01-13 BR BRPI0506777-4A patent/BRPI0506777A/pt not_active Application Discontinuation
- 2005-01-13 JP JP2006549649A patent/JP2007518740A/ja active Pending
- 2005-01-13 CN CNA2005800081262A patent/CN1929844A/zh active Pending
- 2005-01-13 AU AU2005204935A patent/AU2005204935A1/en not_active Abandoned
- 2005-01-13 US US10/585,830 patent/US20080249127A1/en not_active Abandoned
- 2005-01-13 EP EP05711495A patent/EP1711183A4/fr not_active Withdrawn
- 2005-01-13 CA CA002552880A patent/CA2552880A1/fr not_active Abandoned
- 2005-01-13 KR KR1020067016188A patent/KR20060129017A/ko not_active Withdrawn
- 2005-01-13 RU RU2006129289/04A patent/RU2006129289A/ru not_active Application Discontinuation
- 2005-01-13 WO PCT/US2005/001333 patent/WO2005067537A2/fr active Application Filing
-
2006
- 2006-07-10 IL IL176775A patent/IL176775A0/en unknown
- 2006-08-11 NO NO20063636A patent/NO20063636L/no not_active Application Discontinuation
- 2006-08-15 MA MA29273A patent/MA28363A1/fr unknown
Also Published As
Publication number | Publication date |
---|---|
EP1711183A2 (fr) | 2006-10-18 |
US20080249127A1 (en) | 2008-10-09 |
PE20050898A1 (es) | 2005-11-06 |
KR20060129017A (ko) | 2006-12-14 |
TW200534855A (en) | 2005-11-01 |
IL176775A0 (en) | 2006-10-31 |
RU2006129289A (ru) | 2008-02-20 |
AU2005204935A1 (en) | 2005-07-28 |
AR049464A1 (es) | 2006-08-09 |
EP1711183A4 (fr) | 2009-04-01 |
WO2005067537A2 (fr) | 2005-07-28 |
WO2005067537A3 (fr) | 2006-05-18 |
CA2552880A1 (fr) | 2005-07-28 |
JP2007518740A (ja) | 2007-07-12 |
CN1929844A (zh) | 2007-03-14 |
MA28363A1 (fr) | 2006-12-01 |
BRPI0506777A (pt) | 2007-05-22 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FC2A | Withdrawal, rejection or dismissal of laid open patent application |