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WO2006065788A3 - Nouveaux antagonistes du recepteur muscarinique de l'acetylcholine - Google Patents

Nouveaux antagonistes du recepteur muscarinique de l'acetylcholine Download PDF

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Publication number
WO2006065788A3
WO2006065788A3 PCT/US2005/045012 US2005045012W WO2006065788A3 WO 2006065788 A3 WO2006065788 A3 WO 2006065788A3 US 2005045012 W US2005045012 W US 2005045012W WO 2006065788 A3 WO2006065788 A3 WO 2006065788A3
Authority
WO
WIPO (PCT)
Prior art keywords
receptor antagonists
acetylcholine receptor
muscarinic acetylcholine
novel muscarinic
novel
Prior art date
Application number
PCT/US2005/045012
Other languages
English (en)
Other versions
WO2006065788A2 (fr
Inventor
Jakob Busch-Petersen
Roderick S Davis
Wei Fu
Jian Jin
Dramane I Laine
Michael R Palovich
Original Assignee
Glaxo Group Ltd
Jakob Busch-Petersen
Roderick S Davis
Wei Fu
Jian Jin
Dramane I Laine
Michael R Palovich
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd, Jakob Busch-Petersen, Roderick S Davis, Wei Fu, Jian Jin, Dramane I Laine, Michael R Palovich filed Critical Glaxo Group Ltd
Publication of WO2006065788A2 publication Critical patent/WO2006065788A2/fr
Publication of WO2006065788A3 publication Critical patent/WO2006065788A3/fr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

L'invention concerne des antagonistes du récepteur muscarinique de l'acétylcholine, et des méthodes d'utilisation des antagonistes.
PCT/US2005/045012 2004-12-13 2005-12-13 Nouveaux antagonistes du recepteur muscarinique de l'acetylcholine WO2006065788A2 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63570304P 2004-12-13 2004-12-13
US60/635,703 2004-12-13

Publications (2)

Publication Number Publication Date
WO2006065788A2 WO2006065788A2 (fr) 2006-06-22
WO2006065788A3 true WO2006065788A3 (fr) 2006-08-17

Family

ID=36588460

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US2005/045012 WO2006065788A2 (fr) 2004-12-13 2005-12-13 Nouveaux antagonistes du recepteur muscarinique de l'acetylcholine

Country Status (1)

Country Link
WO (1) WO2006065788A2 (fr)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR045914A1 (es) 2003-07-17 2005-11-16 Glaxo Group Ltd Compuesto alcoholico terciario del 8-azoniabiciclo [3.2.1] octano, composicion farmaceutica que lo comprende y su uso para preparar esta ultima
US7276521B2 (en) 2003-10-14 2007-10-02 Glaxo Group Limited Muscarinic acetylcholine receptor antagonists
AU2004281167A1 (en) 2003-10-17 2005-04-28 Glaxo Group Limited Muscarinic acetylcholine receptor antagonists field of the invention
PE20050489A1 (es) 2003-11-04 2005-09-02 Glaxo Group Ltd Antagonistas de receptores de acetilcolina muscarinicos
EP1725564A4 (fr) 2004-03-17 2007-09-12 Glaxo Group Ltd Antagonistes du recepteur d'acetylcholine muscarinique m3
PE20060259A1 (es) 2004-04-27 2006-03-25 Glaxo Group Ltd Compuestos de quinuclidina como antagonistas del receptor de acetilcolina muscarinico
JP2007537261A (ja) 2004-05-13 2007-12-20 グラクソ　グループ　リミテッド ムスカリン性アセチルコリン受容体アンタゴニスト
JP2008520579A (ja) 2004-11-15 2008-06-19 グラクソ グループ リミテッド 新規ｍ３ムスカリン性アセチルコリン受容体アンタゴニスト
WO2006065755A2 (fr) * 2004-12-13 2006-06-22 Glaxo Group Limited Sels d'ammonium quaternaire d'amines heteroaromatiques fusionnees utilises comme nouveaux antagonistes du recepteur de l'acetylcholine muscarinique
EP1937068A4 (fr) 2005-08-18 2010-08-04 Glaxo Group Ltd Antagonistes de recepteurs d'acetylcholine muscarinique
US8188272B2 (en) 2007-03-21 2012-05-29 Bristol-Myers Squibb Company Fused heterocyclic compounds useful as kinase modulators
TW200946525A (en) 2008-02-06 2009-11-16 Glaxo Group Ltd Dual pharmacophores-PDE4-muscarinic antagonistics
TW200946526A (en) 2008-02-06 2009-11-16 Glaxo Group Ltd Dual pharmacophores-PDE4-muscarinic antagonistics
UY31637A1 (es) 2008-02-06 2009-08-03 Farmacoforos duales-antagonistas muscarinicos de pde4
US8476430B2 (en) 2008-07-24 2013-07-02 Bristol-Myers Squibb Company Fused heterocyclic compounds useful as kinase modulators
WO2010094643A1 (fr) 2009-02-17 2010-08-26 Glaxo Group Limited Dérivés de quinoline et applications associées dans la rhinite et l'urticaire
GB0918924D0 (en) * 2009-10-28 2009-12-16 Vantia Ltd Azaindole derivatives
TW201414737A (zh) 2012-07-13 2014-04-16 必治妥美雅史谷比公司 作爲激酶抑制劑之咪唑并三□甲腈

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6657064B2 (en) * 1999-10-08 2003-12-02 Gruenenthal Gmbh Bicyclic imidazo-5-yl-amine derivatives

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6657064B2 (en) * 1999-10-08 2003-12-02 Gruenenthal Gmbh Bicyclic imidazo-5-yl-amine derivatives

Also Published As

Publication number Publication date
WO2006065788A2 (fr) 2006-06-22

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