SE8800613D0
(sv)
|
1988-02-23 |
1988-02-23 |
Wallac Oy |
A novel spectrofluorometric method and compounds that are of value for the method
|
JPH03287584A
(ja)
|
1990-04-05 |
1991-12-18 |
Banyu Pharmaceut Co Ltd |
置換アリルアミン誘導体
|
US5250534A
(en)
|
1990-06-20 |
1993-10-05 |
Pfizer Inc. |
Pyrazolopyrimidinone antianginal agents
|
US6200980B1
(en)
|
1995-06-07 |
2001-03-13 |
Cell Pathways, Inc. |
Method of treating a patient having precancerous lesions with phenyl purinone derivatives
|
IL132276A0
(en)
|
1997-04-25 |
2001-03-19 |
Pfizer |
Pyrazolopyrimidinones which inhibit type 5 cyclic guanosine 3',5'-monophosphate phosphodiesterase (cgmp pde5) for the treatment of sexual dysfunction
|
AU748352B2
(en)
|
1998-04-20 |
2002-06-06 |
Pfizer Inc. |
Pyrazolopyrimidinone cGMP PDE5 inhibitors for the treatment of sexual dysfunction
|
JP2000038350A
(ja)
|
1998-05-18 |
2000-02-08 |
Yoshitomi Pharmaceut Ind Ltd |
糖尿病治療薬
|
GB9823101D0
(en)
|
1998-10-23 |
1998-12-16 |
Pfizer Ltd |
Pharmaceutically active compounds
|
GB9823102D0
(en)
|
1998-10-23 |
1998-12-16 |
Pfizer Ltd |
Pharmaceutically active compounds
|
WO2001046124A1
(fr)
|
1999-12-22 |
2001-06-28 |
Nihon Nohyaku Co., Ltd. |
Derives de diamide aromatique, produits chimiques utilises en agriculture ou en horticulture et utilisations de ces derniers
|
CZ27399A3
(cs)
|
1999-01-26 |
2000-08-16 |
Ústav Experimentální Botaniky Av Čr |
Substituované dusíkaté heterocyklické deriváty, způsob jejich přípravy, tyto deriváty pro použití jako léčiva, farmaceutická kompozice a kombinovaný farmaceutický přípravek tyto deriváty obsahující a použití těchto derivátů pro výrobu léčiv
|
IN187433B
(fr)
|
1999-09-10 |
2002-04-27 |
Cipla Ltd |
|
AU1888800A
(en)
|
1999-09-13 |
2001-04-17 |
Cipla Limited |
A novel process for the synthesis of sildenafil citrate
|
CZ2002934A3
(cs)
|
1999-09-17 |
2002-07-17 |
Abbott Gmbh & Co. Kg |
Inhibitory kinázy jako terapeutická činidla
|
US6864289B1
(en)
|
1999-09-24 |
2005-03-08 |
Nihon Nohyaku Co., Ltd. |
Aromatic diamide derivatives or salts thereof, agricultural/horticultural chemicals and method of using the same
|
TR200200954T2
(tr)
|
1999-10-11 |
2002-09-23 |
Pfizer Inc. |
Fosfodiesteraz inhibitörleri olarak 5-(2-ikame edilmiş-5-heterosiklilsülfonilpirid-3-il)- dihidropirazolo[4,3- D]pirimidin-7-onlar.
|
TWI265925B
(en)
|
1999-10-11 |
2006-11-11 |
Pfizer |
Pyrazolo[4,3-d]pyrimidin-7-ones useful in inhibiting type 5 cyclic guanosine 3',5'-monophosphate phosphodiesterases(cGMP PDE5), process and intermediates for their preparation, their uses and composition comprising them
|
IL152925A
(en)
|
1999-10-21 |
2010-04-15 |
Pfizer |
Pharmaceutical preparations for the treatment of neurological disease containing an inhibitor of ring guanizine '3', 5 '- monophosphate phosphodiesterase 5 and one of gabapentin or pregabalin
|
MXPA99010322A
(es)
|
1999-11-10 |
2003-07-15 |
Europharm S A De C V |
Proceso para la preparacion de sildenafil.
|
CO5271697A1
(es)
|
2000-01-12 |
2003-04-30 |
Pfizer Prod Inc |
Composiciones y procedimientos para el tratamiento de afecciones que responden a un aumento de testosterona
|
US20020013327A1
(en)
|
2000-04-18 |
2002-01-31 |
Lee Andrew G. |
Compositions and methods for treating female sexual dysfunction
|
PL202623B1
(pl)
|
2000-06-28 |
2009-07-31 |
Smithkline Beecham Plc |
Sposób wytwarzania drobno zmielonego preparatu substancji leczniczej, drobno zmielona substancja lecznicza wytworzona tym sposobem i zawierająca ją kompozycja farmaceutyczna
|
AU2001277621A1
(en)
|
2000-08-09 |
2002-03-04 |
Astrazeneca Ab |
Antiangiogenic bicyclic derivatives
|
AU2001284417A1
(en)
|
2000-09-05 |
2002-03-22 |
Taisho Pharmaceutical Co. Ltd. |
Hair growth stimulants
|
US6548508B2
(en)
|
2000-10-20 |
2003-04-15 |
Pfizer, Inc. |
Use of PDE V inhibitors for improved fecundity in mammals
|
JP2004518662A
(ja)
|
2000-12-19 |
2004-06-24 |
スミスクライン ビーチャム パブリック リミテッド カンパニー |
Gsk−3阻害剤としてのピラゾロ[3,4−c]ピリジン
|
CA2431077A1
(fr)
|
2000-12-19 |
2002-06-27 |
Merck Patent Gesellschaft Mit Beschraenkter Haftung |
Formulation pharmaceutique contenant des pyrazolo[4,3-d]pyrimidines et des antithrombotiques, des antagonistes de calcium, des prostaglandines ou des derives de prostaglandine
|
US6770645B2
(en)
|
2001-03-16 |
2004-08-03 |
Pfizer Inc. |
Pharmaceutically active compounds
|
US6784185B2
(en)
|
2001-03-16 |
2004-08-31 |
Pfizer Inc. |
Pharmaceutically active compounds
|
US7902179B2
(en)
|
2001-04-26 |
2011-03-08 |
Ajinomoto Co., Inc. |
Heterocyclic compounds
|
EP1383760A1
(fr)
|
2001-04-30 |
2004-01-28 |
Fujisawa Pharmaceutical Co., Ltd. |
Composes biarylcarboxamide comme inhibiteurs d'apolipoproteine b
|
FR2825706B1
(fr)
|
2001-06-06 |
2003-12-12 |
Pf Medicament |
Nouveaux derives de benzothienyle ou d'indole, leur preparation et leur utilisation comme inhibiteurs de proteines prenyl transferase
|
IL161155A0
(en)
|
2001-11-02 |
2004-08-31 |
Pfizer Prod Inc |
Treatment of insulin resistance syndrome and type 2 diabetes with pde9 inhibitors
|
TW200738672A
(en)
|
2001-12-10 |
2007-10-16 |
Bristol Myers Squibb Co |
Intermediated for the preparation of 4,5-dihydro-pyrazolo [3,4-c] pyrid-2-ones
|
US7166293B2
(en)
|
2002-03-29 |
2007-01-23 |
Carlsbad Technology, Inc. |
Angiogenesis inhibitors
|
US20050119278A1
(en)
|
2002-05-16 |
2005-06-02 |
Che-Ming Teng |
Anti-angiogenesis methods
|
EP1510516A4
(fr)
|
2002-05-31 |
2005-11-02 |
Eisai Co Ltd |
Compose de pyrazole et composition medicinale le contenant
|
ES2337254T3
(es)
|
2003-02-14 |
2010-04-22 |
Glaxo Group Limited |
Derivados de carboxamida.
|
WO2004074286A1
(fr)
|
2003-02-14 |
2004-09-02 |
Wyeth |
Derives de heterocyclyl-3-sulfonylazaindole ou -azaindazole utilises comme ligands de la 5-hydroxytryptamine-6
|
EP1613747A1
(fr)
|
2003-03-31 |
2006-01-11 |
Pfizer Products Inc. |
Structure cristalline de 3',5'-phosphodiesterase nucleotidique cyclique 1d(pde1b) et ses utilisations
|
WO2004096810A1
(fr)
|
2003-04-29 |
2004-11-11 |
Pfizer Limited |
5,7-diaminopyrazolo`4,3-d!pyrimidines utiles pour le traitement de l'hypertension
|
EP1628661A2
(fr)
|
2003-06-05 |
2006-03-01 |
Vertex Pharmaceuticals Incorporated |
Modulateurs du recepteur vr1
|
EP1635812A2
(fr)
|
2003-06-10 |
2006-03-22 |
Fulcrum Pharmaceuticals, Inc. |
Inhibiteurs de beta-lactamases et methodes d'utilisation de ces inhibiteurs
|
ZA200305330B
(en)
|
2003-07-10 |
2004-05-26 |
Jb Chemicals & Pharmaceuticals |
An improved process for the preparation of 5-[2-ethoxy-5-(4-methylpiperazin-1-ylsulphonyl)phenyl]-1-methyl-3-n-propyl-1,6-dihydro-7H-pyrazole[4,3-D]P yrimidin-7-one.
|
EP1648448A4
(fr)
|
2003-07-29 |
2009-04-01 |
Smithkline Beecham Corp |
Composes chimiques
|
TWI339206B
(en)
|
2003-09-04 |
2011-03-21 |
Vertex Pharma |
Compositions useful as inhibitors of protein kinases
|
PL1689233T3
(pl)
|
2003-11-19 |
2012-11-30 |
Array Biopharma Inc |
Bicykliczne inhibitory MEK
|
US20050137398A1
(en)
|
2003-12-22 |
2005-06-23 |
Jianguo Ji |
3-Quinuclidinyl heteroatom bridged biaryl derivatives
|
US7241773B2
(en)
|
2003-12-22 |
2007-07-10 |
Abbott Laboratories |
3-quinuclidinyl heteroatom bridged biaryl derivatives
|
GB0402137D0
(en)
|
2004-01-30 |
2004-03-03 |
Smithkline Beecham Corp |
Novel compounds
|
DE102004005172A1
(de)
|
2004-02-02 |
2005-08-18 |
Aventis Pharma Deutschland Gmbh |
Indazolderivate als Inhibitoren der Hormon Sensitiven Lipase
|
RU2006134021A
(ru)
|
2004-02-27 |
2008-04-10 |
Ф.Хоффманн-Ля Рош Аг (Ch) |
Производные гетероарил-конденсированного пиразола
|
KR100843526B1
(ko)
|
2004-02-27 |
2008-07-03 |
에프. 호프만-라 로슈 아게 |
피라졸의 접합 유도체
|
JP2007526324A
(ja)
|
2004-03-02 |
2007-09-13 |
スミスクライン・ビーチャム・コーポレイション |
Akt活性のある阻害剤
|
AR050188A1
(es)
|
2004-08-03 |
2006-10-04 |
Uriach Y Compania S A J |
Compuestos heterociclicos condensados utiles en terapia como inhibidores de quinasas p38 y composiciones farmaceuticas que los contienen
|
EA201890903A9
(ru)
|
2004-09-02 |
2021-11-10 |
Дженентек, Инк. |
Соединения пиридиловых ингибиторов передачи сигналов белком hedgehog, способ их получения, композиция и способы лечения рака и ингибирований ангиогенеза и сигнального пути hedgehog в клетках на их основе
|
WO2006038001A1
(fr)
|
2004-10-06 |
2006-04-13 |
Celltech R & D Limited |
Derives d’aminopyrimidine en tant qu’inhibiteurs de la jnk
|
CA2584485C
(fr)
|
2004-10-20 |
2013-12-31 |
Resverlogix Corp. |
Stilbenes et chalcones utilises pour la prevention et le traitement de maladies cardio-vasculaires
|
AR051596A1
(es)
|
2004-10-26 |
2007-01-24 |
Irm Llc |
Compuestos heterociclicos condensados nitrogenados como inhibidores de la actividad del receptor canabinoide 1; composiciones farmaceuticas que los contienen y su empleo en la preparacion de medicamentos para el tratamiento de trastornos alimentarios
|
TW200630327A
(en)
|
2004-10-28 |
2006-09-01 |
Inst For Pharm Discovery Inc |
Substituted phenylalkanoic acids
|
CA2586870A1
(fr)
|
2004-11-10 |
2006-05-18 |
Synta Pharmaceuticals Corp. |
Composes modulateurs de la il-12
|
US7919487B2
(en)
|
2004-11-10 |
2011-04-05 |
Synta Pharmaceuticals Corporation |
Heteroaryl compounds
|
EP1812442A2
(fr)
|
2004-11-10 |
2007-08-01 |
CGI Pharmaceuticals, Inc. |
Certaines imidazo[1,2-a] pyrazin-8-ylamines et les procédés de fabrication et d'utilisation correspondants
|
DE102004054666A1
(de)
|
2004-11-12 |
2006-05-18 |
Bayer Cropscience Gmbh |
Substituierte Pyrazol-3-carboxamide, Verfahren zur Herstellung und Verwendung als Herbizide und Pflanzenwachstumsregulatoren
|
CN100516049C
(zh)
|
2004-11-16 |
2009-07-22 |
永信药品工业股份有限公司 |
抗血管生成药n2-(取代的芳基甲基)-3-(取代的苯基)吲唑的合成
|
WO2006074428A2
(fr)
|
2005-01-07 |
2006-07-13 |
Emory University |
Antagonistes de cxcr4 pour le traitement de troubles medicaux
|
EP1863483A4
(fr)
|
2005-03-31 |
2010-03-31 |
Janssen Pharmaceutica Nv |
Composes de pyrazole bicycliques utilises comme agents antibacteriens
|
US20070032493A1
(en)
|
2005-05-26 |
2007-02-08 |
Synta Pharmaceuticals Corp. |
Method for treating B cell regulated autoimmune disorders
|
US20100216798A1
(en)
|
2005-07-29 |
2010-08-26 |
Astellas Pharma Inc |
Fused heterocycles as lck inhibitors
|
JP5203196B2
(ja)
|
2005-08-04 |
2013-06-05 |
サートリス ファーマシューティカルズ, インコーポレイテッド |
サーチュインモジュレーターとしてのオキサゾロピリジン誘導体
|
GB0516703D0
(en)
|
2005-08-15 |
2005-09-21 |
Syngenta Participations Ag |
Novel insecticides
|
JP2007055940A
(ja)
|
2005-08-24 |
2007-03-08 |
Astellas Pharma Inc |
ピラゾロピリミジン誘導体
|
CN101243051A
(zh)
|
2005-08-25 |
2008-08-13 |
霍夫曼-拉罗奇有限公司 |
p38 MAP激酶抑制剂及使用它的方法
|
JP2009506007A
(ja)
|
2005-08-25 |
2009-02-12 |
エフ.ホフマン−ラ ロシュ アーゲー |
p38MAPキナーゼ阻害剤及びその使用方法
|
CN101243090A
(zh)
|
2005-08-25 |
2008-08-13 |
霍夫曼-拉罗奇有限公司 |
p38 MAP激酶抑制剂及使用它的方法
|
EP1922311A2
(fr)
|
2005-09-09 |
2008-05-21 |
Brystol-Myers Squibb Company |
Inhibiteurs d'ikur acycliques
|
WO2007041511A2
(fr)
|
2005-09-30 |
2007-04-12 |
New York University |
Kinase des progeniteurs hematopoietiques 1 destinee a la modulation d'une reponse immune
|
US20080242685A1
(en)
*
|
2005-10-25 |
2008-10-02 |
Smithkline Beecham Corporation |
Chemical Compounds
|
EP1948604A1
(fr)
|
2005-11-03 |
2008-07-30 |
Ilypsa, Inc. |
Composes d'indole presentant des substituants acides c4 et leur utilisation en tant qu'inhibiteurs de phospholipases a2
|
KR20080071562A
(ko)
|
2005-11-30 |
2008-08-04 |
아스텔라스세이야쿠 가부시키가이샤 |
2-아미노벤즈아미드 유도체
|
GB0525143D0
(en)
|
2005-12-09 |
2006-01-18 |
Novartis Ag |
Organic compounds
|
AU2007204208A1
(en)
|
2006-01-11 |
2007-07-19 |
Astrazeneca Ab |
Morpholino pyrimidine derivatives and their use in therapy
|
TW200808766A
(en)
|
2006-02-16 |
2008-02-16 |
Syngenta Participations Ag |
Novel insecticides
|
WO2007112093A2
(fr)
|
2006-03-23 |
2007-10-04 |
Synta Pharmaceuticals Corp. |
Composés de benzimidazolyl-pyridine pour le traitement de l'inflammation et de troubles immunitaires
|
MX2008012400A
(es)
|
2006-03-30 |
2008-10-10 |
Irm Llc |
Azolopirimidinas como inhibidores de actividad de cannabinoide 1.
|
NZ573735A
(en)
|
2006-05-19 |
2011-10-28 |
Abbott Lab |
Cns active fused bicycloheterocycle substituted azabicyclic alkane derivatives
|
US20080280891A1
(en)
|
2006-06-27 |
2008-11-13 |
Locus Pharmaceuticals, Inc. |
Anti-cancer agents and uses thereof
|
WO2008008059A1
(fr)
|
2006-07-12 |
2008-01-17 |
Locus Pharmaceuticals, Inc. |
Agents anti-cancer et leurs utilisations
|
PE20121506A1
(es)
|
2006-07-14 |
2012-11-26 |
Amgen Inc |
Compuestos triazolopiridinas como inhibidores de c-met
|
GB0614691D0
(en)
|
2006-07-24 |
2006-08-30 |
Syngenta Participations Ag |
Insecticidal compounds
|
MX2009003649A
(es)
|
2006-10-06 |
2009-04-22 |
Irm Llc |
Inhibidores de cinasa de proteina y metodos para utilizarlos.
|
MX2009003941A
(es)
|
2006-10-20 |
2009-04-24 |
Concert Pharmaceuticals Inc |
Derivados de 3-(dihidro-1h-pirazolo[4,3-d]pirimidin-5-il)-4-propox ibencenosulfonamida y metodos de uso.
|
US20080194557A1
(en)
|
2007-01-18 |
2008-08-14 |
Joseph Barbosa |
Methods and compositions for the treatment of pain, inflammation and cancer
|
WO2008089310A2
(fr)
|
2007-01-18 |
2008-07-24 |
Lexicon Pharmaceuticals, Inc. |
Méthodes et compositions utilisées dans le traitement de troubles corporels
|
US20140249135A1
(en)
|
2007-03-01 |
2014-09-04 |
Novartis Ag |
Pim kinase inhibitors and methods of their use
|
EP2002835A1
(fr)
|
2007-06-04 |
2008-12-17 |
GenKyo Tex |
Dérivés de pyrazolo pyridine en tant qu'inhibiteurs de la NADPH oxydase
|
MY146643A
(en)
|
2007-07-30 |
2012-09-14 |
Dae Woong Pharma |
Novel benzoimidazole derivatives and pharmaceutical composition comprising the same
|
CN101790519B
(zh)
|
2007-08-08 |
2013-10-16 |
默克雪兰诺有限公司 |
用于治疗多发性硬化症的结合于鞘氨醇1-磷酸(s1p)的6-氨基-嘧啶-4-羧酰胺衍生物及相关化合物
|
GB0716414D0
(en)
|
2007-08-22 |
2007-10-03 |
Syngenta Participations Ag |
Novel insecticides
|
WO2009032651A1
(fr)
|
2007-08-31 |
2009-03-12 |
Smithkline Beecham Corporation |
INHIBITEURS DE L'ACTIVITÉ Akt
|
US8314131B2
(en)
|
2007-09-21 |
2012-11-20 |
Amgen Inc. |
Triazole fused heteroaryl compounds and methods of use thereof
|
BRPI0819093A2
(pt)
|
2007-11-01 |
2017-05-02 |
Sirtris Pharmaceuticals Inc |
compostos moduladores de sirtuína
|
KR100963644B1
(ko)
|
2007-11-23 |
2010-06-15 |
한국과학기술연구원 |
피라졸로피리미딘온 유도체 및 그의 제조방법
|
UA106037C2
(uk)
|
2008-02-04 |
2014-07-25 |
Мерк'Юрі Терап'Ютікс, Інк. |
Модулятори ampk (амф-активованої протеїнкінази)
|
US20110124634A1
(en)
|
2008-05-13 |
2011-05-26 |
Poniard Pharmaceuticals, Inc. |
Bioactive compounds for treatment of cancer and neurodegenerative diseases
|
CN102089278A
(zh)
|
2008-06-11 |
2011-06-08 |
Irm责任有限公司 |
用于治疗疟疾的化合物和组合物
|
EP2361248B1
(fr)
|
2008-06-27 |
2018-09-19 |
Celgene CAR LLC |
Composés hétéro-aryles et leurs utilisations
|
US20110294853A1
(en)
|
2008-09-12 |
2011-12-01 |
Benjamin Pelcman |
Bis Aromatic Compounds for Use in the Treatment of Inflammation
|
EP2166008A1
(fr)
|
2008-09-23 |
2010-03-24 |
Genkyo Tex Sa |
Dérivés de pyridine pyrazolo en tant qu'inhibiteurs d'oxydase NADPH
|
EP2166010A1
(fr)
|
2008-09-23 |
2010-03-24 |
Genkyo Tex Sa |
Dérivés de pyridine pyrazolo en tant qu'inhibiteurs d'oxydase NADPH
|
EP2165707A1
(fr)
|
2008-09-23 |
2010-03-24 |
Genkyo Tex Sa |
Dérivés de pyrazolo pyridine en tant qu'inhibiteurs de la NADPH oxydase
|
WO2010046780A2
(fr)
|
2008-10-22 |
2010-04-29 |
Institut Pasteur Korea |
Composés antiviraux
|
JP2010111624A
(ja)
|
2008-11-06 |
2010-05-20 |
Shionogi & Co Ltd |
Ttk阻害作用を有するインダゾール誘導体
|
ES2544452T3
(es)
|
2008-12-19 |
2015-08-31 |
Genentech, Inc. |
Compuestos heterocíclicos y métodos de uso
|
KR20100101056A
(ko)
|
2009-03-07 |
2010-09-16 |
주식회사 메디젠텍 |
세포핵에서 세포질로의 gsk3의 이동을 억제하는 화합물을 함유하는 세포핵에서 세포질로의 gsk3 이동에 의해 발생되는 질환의 치료 또는 예방용 약학적 조성물
|
EP2408744A1
(fr)
|
2009-03-18 |
2012-01-25 |
Schering Corporation |
Composés bicycliques en tant qu'inhibiteurs de la diacylglycérol acyltransférase
|
EP3584217B1
(fr)
|
2009-03-26 |
2023-07-05 |
Northeastern University |
Nanostructures de carbone provenant de la pyrolyse de matières organiques
|
WO2010118367A2
(fr)
|
2009-04-10 |
2010-10-14 |
Progenics Pharmaceuticals, Inc. |
Pyrimidines antivirales
|
WO2011019780A1
(fr)
|
2009-08-11 |
2011-02-17 |
Bristol-Myers Squibb Company |
Azaindazoles comme modulateurs de la kinase btk et leur utilisation
|
EP2477498A4
(fr)
|
2009-09-14 |
2013-02-27 |
Merck Sharp & Dohme |
Inhibiteurs de diacylglycérol acyltransférase
|
WO2011050245A1
(fr)
|
2009-10-23 |
2011-04-28 |
Yangbo Feng |
Hétéroaryles bicycliques formant inhibiteurs de la kinase
|
ES2360333B1
(es)
|
2009-10-29 |
2012-05-04 |
Consejo Superior De Investigaciones Cientificas (Csic) (70%) |
Derivados de bis (aralquil) amino y sistemas (hetero) aromaticos de seis miembros y su uso en el tratamiento de patologias neurodegenerativas, incluida la enfermedad de alzheimer
|
JP2013032290A
(ja)
|
2009-11-20 |
2013-02-14 |
Dainippon Sumitomo Pharma Co Ltd |
新規縮合ピリミジン誘導体
|
WO2011078143A1
(fr)
|
2009-12-22 |
2011-06-30 |
塩野義製薬株式会社 |
Dérivés de pyrimidine et composition pharmaceutique les contenant
|
US9180127B2
(en)
|
2009-12-29 |
2015-11-10 |
Dana-Farber Cancer Institute, Inc. |
Type II Raf kinase inhibitors
|
WO2011082400A2
(fr)
|
2010-01-04 |
2011-07-07 |
President And Fellows Of Harvard College |
Modulateurs du récepteur immunosuppresseur pd-1 et procédés d'utilisation de ceux-ci
|
AR079975A1
(es)
|
2010-01-06 |
2012-03-07 |
British Columbia Cancer Agency |
Agentes terapeuticos derivados de bisfenol u metodos para su uso, composiciones farmaceuticas y uso de los mismos
|
DE102010009903A1
(de)
|
2010-03-02 |
2011-09-08 |
Merck Patent Gmbh |
Verbindungen für elektronische Vorrichtungen
|
CN102206172B
(zh)
|
2010-03-30 |
2015-02-25 |
中国医学科学院医药生物技术研究所 |
一组取代双芳基化合物及其制备方法和抗病毒应用
|
EP2560488B1
(fr)
|
2010-04-23 |
2015-10-28 |
Cytokinetics, Inc. |
Aminopyridines et aminotriazines, leurs compositions et leurs procédés d'utilisation
|
PL2563776T3
(pl)
|
2010-04-27 |
2017-01-31 |
Calcimedica Inc |
Związki, które modulują wewnątrzkomórkowy wapń
|
GB201008134D0
(en)
|
2010-05-14 |
2010-06-30 |
Medical Res Council Technology |
Compounds
|
JP2011246389A
(ja)
|
2010-05-26 |
2011-12-08 |
Oncotherapy Science Ltd |
Ttk阻害作用を有する縮環ピラゾール誘導体
|
BR112012030184A2
(pt)
|
2010-05-27 |
2015-12-29 |
Bayer Cropscience Ag |
derivados de ácido piridinilcarboxílico como fungicidas
|
WO2011153553A2
(fr)
|
2010-06-04 |
2011-12-08 |
The Regents Of The University Of California |
Méthodes et compositions pour l'inhibition de kinases
|
JP5993846B2
(ja)
|
2010-06-15 |
2016-09-14 |
バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH |
アントラニル酸誘導体
|
US9212139B2
(en)
|
2010-06-16 |
2015-12-15 |
Purdue Pharma, L.P. |
Aryl substituted indoles and their use as blockers of sodium channels
|
JP5926727B2
(ja)
|
2010-07-28 |
2016-05-25 |
バイエル・インテレクチュアル・プロパティ・ゲゼルシャフト・ミット・ベシュレンクテル・ハフツングBayer Intellectual Property GmbH |
置換イミダゾ[1,2−b]ピリダジン
|
WO2012048058A2
(fr)
|
2010-10-06 |
2012-04-12 |
J-Pharma Co., Ltd. |
Développement de puissants inhibiteurs des transporteurs d'urate : composés conçus pour leur action uricosurique
|
GB201017345D0
(en)
|
2010-10-14 |
2010-11-24 |
Proximagen Ltd |
Receptor antagonists
|
WO2012078777A1
(fr)
|
2010-12-09 |
2012-06-14 |
Amgen Inc. |
Composés bicycliques en tant qu'inhibiteurs de pim
|
US20130253011A1
(en)
|
2010-12-17 |
2013-09-26 |
Syngenta Participations Ag |
Insecticidal compounds
|
JP5921572B2
(ja)
|
2011-01-04 |
2016-05-24 |
ノバルティス アーゲー |
加齢性黄斑変性症(amd)の処置に有用なインドール化合物またはそのアナログ
|
ES2732311T3
(es)
|
2011-02-07 |
2019-11-21 |
Univ Washington |
Compuestos de manósidos y procedimientos de uso de los mismos
|
EP2691399B1
(fr)
|
2011-03-28 |
2016-07-13 |
F.Hoffmann-La Roche Ag |
Composés thiazolopyrimidines
|
PL2697207T3
(pl)
|
2011-04-12 |
2017-08-31 |
Chong Kun Dang Pharmaceutical Corp. |
Pochodne 3-(2-arylocykloalkenylometylo)oksazolidyn-2-onu jako inhibitory białka transportującego estry cholesterolu (cetp)
|
MX363696B
(es)
|
2011-04-21 |
2019-03-28 |
Origenis Gmbh |
Pirazolo[4,3-d]pirimidinas utiles como inhibidores de cinasas.
|
US20140288069A1
(en)
|
2011-05-17 |
2014-09-25 |
Bayer Intellectual Property Gmbh |
Amino-substituted imidazopyridazines as mknk1 kinase inhibitors
|
WO2012158810A1
(fr)
|
2011-05-17 |
2012-11-22 |
Principia Biopharma Inc. |
Inhibiteurs de tyrosine kinase
|
UY34104A
(es)
|
2011-05-31 |
2013-01-03 |
Syngenta Participations Ag |
?compuestos derivados benzamídicos heterocíclicos, procesos e intermedios para su preparación, composiciones y métodos para su uso?.
|
WO2012163942A1
(fr)
|
2011-06-01 |
2012-12-06 |
Bayer Intellectual Property Gmbh |
Aminoimidazopyridazines substituées
|
EP2723748B1
(fr)
|
2011-06-22 |
2016-10-12 |
Bayer Intellectual Property GmbH |
Hétérocyclylaminoimidazopyridazines
|
EP2543372A1
(fr)
|
2011-07-08 |
2013-01-09 |
Helmholtz-Zentrum für Infektionsforschung GmbH |
Médicament pour le traitement du cancer du foie
|
EP3111937B1
(fr)
|
2011-07-08 |
2020-06-17 |
Helmholtz-Zentrum für Infektionsforschung GmbH |
Médicament pour le traitement du cancer du foie
|
AU2012293417A1
(en)
|
2011-08-10 |
2013-05-02 |
Purdue Pharma L.P. |
TRPV1 antagonists including dihydroxy substituent and uses thereof
|
WO2013024002A1
(fr)
|
2011-08-12 |
2013-02-21 |
F. Hoffmann-La Roche Ag |
Composés de pyrazolo[3,4-c]pyridine et procédés d'utilisation
|
RU2014105624A
(ru)
|
2011-08-12 |
2015-09-20 |
Ф. Хоффманн-Ля Рош Аг |
Соединения индазола, способ их применения и фармацевтическая композиция
|
WO2013042137A1
(fr)
|
2011-09-19 |
2013-03-28 |
Aurigene Discovery Technologies Limited |
Hétérocycles bicycliques convenant comme inhibiteurs de l'irak4
|
CN103814029B
(zh)
|
2011-09-23 |
2016-10-12 |
拜耳知识产权有限责任公司 |
取代的咪唑并哒嗪
|
CN102516263B
(zh)
|
2011-10-25 |
2015-04-08 |
南方医科大学 |
一种螺三环类化合物及其制备方法、以及含该类化合物的药物组合物及其应用
|
CN102503959B
(zh)
|
2011-10-25 |
2015-04-08 |
南方医科大学 |
一种稠三环类化合物及其制备方法、以及含该类化合物的药物组合物及其应用
|
WO2013064445A1
(fr)
|
2011-11-01 |
2013-05-10 |
F. Hoffmann-La Roche Ag |
Composés d'imidazopyridazine
|
JP6200903B2
(ja)
|
2012-02-17 |
2017-09-20 |
キネタ フォー エルエルシー |
アレナウイルス感染症の治療のための抗ウイルス薬
|
TW201348231A
(zh)
|
2012-02-29 |
2013-12-01 |
Amgen Inc |
雜雙環化合物
|
CN104169260A
(zh)
|
2012-03-09 |
2014-11-26 |
卡尔那生物科学株式会社 |
新三嗪衍生物
|
JP6101248B2
(ja)
|
2012-03-28 |
2017-03-22 |
出光興産株式会社 |
新規化合物、有機エレクトロルミネッセンス素子用材料および有機エレクトロルミネッセンス素子
|
ES2571479T3
(es)
|
2012-04-20 |
2016-05-25 |
Gilead Sciences Inc |
Derivados del ácido benzotiazol-6-il acético y su uso para tratar una infección por VIH
|
WO2014003405A1
(fr)
|
2012-06-26 |
2014-01-03 |
주식회사 제이앤드제이 캐미칼 |
Nouveau composé et dispositif émettant de la lumière le comprenant
|
CA2876993A1
(fr)
|
2012-06-28 |
2014-01-03 |
Novartis Ag |
Derives de pyrrolidine et leur utilisation en tant que modulateurs des voies du complement
|
KR101936851B1
(ko)
|
2012-07-16 |
2019-01-11 |
한국과학기술연구원 |
단백질 키나아제 저해제인 신규 피라졸로피리딘 유도체 또는 인다졸 유도체
|
WO2014024125A1
(fr)
|
2012-08-08 |
2014-02-13 |
Celon Pharma S.A. |
Dérivés pyrazolo[4,3-d]pyrimidin-7(6h)-one comme inhibiteurs de pde9
|
JPWO2014030716A1
(ja)
|
2012-08-23 |
2016-08-08 |
田辺三菱製薬株式会社 |
ピラゾロピリミジン化合物
|
US9882150B2
(en)
|
2012-09-24 |
2018-01-30 |
Arizona Board Of Regents For And On Behalf Of Arizona State University |
Metal compounds, methods, and uses thereof
|
EP2903978B1
(fr)
|
2012-10-05 |
2022-12-07 |
Rigel Pharmaceuticals, Inc. |
Inhibiteurs de gdf-8
|
KR102137472B1
(ko)
|
2013-02-08 |
2020-07-27 |
삼성디스플레이 주식회사 |
유기 발광 소자
|
US9242969B2
(en)
|
2013-03-14 |
2016-01-26 |
Novartis Ag |
Biaryl amide compounds as kinase inhibitors
|
WO2014152013A1
(fr)
|
2013-03-14 |
2014-09-25 |
The Trustees Of Columbia University In The City Of New York |
4-phénylpipéridines, leur préparation et leur utilisation
|
US9227978B2
(en)
|
2013-03-15 |
2016-01-05 |
Araxes Pharma Llc |
Covalent inhibitors of Kras G12C
|
US9034927B2
(en)
|
2013-05-22 |
2015-05-19 |
Curza Global, Llc |
Methods of use for compositions comprising a biocidal polyamine
|
JP6603445B2
(ja)
|
2013-06-10 |
2019-11-06 |
アリゾナ・ボード・オブ・リージェンツ・オン・ビハーフ・オブ・アリゾナ・ステイト・ユニバーシティー |
改変された発光スペクトルを有する蛍光性四座配位金属錯体
|
WO2015026683A1
(fr)
*
|
2013-08-22 |
2015-02-26 |
Merck Sharp & Dohme Corp. |
Composés inhibant l'activité enzymatique de la kinase à répétitions riches en leucine
|
TWI652014B
(zh)
|
2013-09-13 |
2019-03-01 |
美商艾佛艾姆希公司 |
雜環取代之雙環唑殺蟲劑
|
WO2015037965A1
(fr)
|
2013-09-16 |
2015-03-19 |
Rohm And Haas Electronic Materials Korea Ltd. |
Nouveaux composés électroluminescents organiques et dispositif électroluminescent organique les comprenant
|
WO2015058163A2
(fr)
|
2013-10-18 |
2015-04-23 |
Syros Pharmaceuticals, Inc. |
Inhibiteurs de la kinase cycline-dépendante 7 (cdk7)
|
MX2016005054A
(es)
|
2013-10-21 |
2016-07-19 |
Merck Patent Gmbh |
Compuestos heteroarilo como inhibidores de tirosina cinasa de bruton (bkt) y usos de los mismos.
|
EP3444251B1
(fr)
|
2013-12-11 |
2023-06-07 |
Biogen MA Inc. |
Composés biaryles utiles dans le traitement de maladies humaines en oncologie, neurologie et immunologie
|
US9856223B2
(en)
*
|
2013-12-13 |
2018-01-02 |
Dana-Farber Cancer Institute, Inc. |
Methods to treat lymphoplasmacytic lymphoma
|
TWI667233B
(zh)
|
2013-12-19 |
2019-08-01 |
德商拜耳製藥公司 |
新穎吲唑羧醯胺,其製備方法、含彼等之醫藥製劑及其製造醫藥之用途
|
EP3083589B1
(fr)
|
2013-12-20 |
2019-12-18 |
Sunshine Lake Pharma Co., Ltd. |
Composés pipéraziniques substitués et leurs procédés d'utilisation
|
KR20160115933A
(ko)
|
2014-01-10 |
2016-10-06 |
오리진 디스커버리 테크놀로지스 리미티드 |
Irak4 억제제로서의 인다졸 화합물
|
WO2015117718A1
(fr)
|
2014-02-05 |
2015-08-13 |
Merck Patent Gmbh |
Complexes métalliques
|
KR20160116018A
(ko)
|
2014-02-25 |
2016-10-06 |
아칠리온 파르마세우티칼스 인코포레이티드 |
보체 매개 질환의 치료를 위한 아미드 화합물
|
US9871208B2
(en)
|
2014-02-26 |
2018-01-16 |
Samsung Display Co., Ltd. |
Condensed cyclic compound and organic light-emitting device including the same
|
WO2015164956A1
(fr)
|
2014-04-29 |
2015-11-05 |
The University Of British Columbia |
Composés dérivés de benzisothiazole utilisés comme agents thérapeutiques et leurs méthodes d'utilisation
|
US20150328188A1
(en)
|
2014-05-19 |
2015-11-19 |
Everardus O. Orlemans |
Combination Therapies for the Treatment of Proliferative Disorders
|
EP3158597B1
(fr)
|
2014-06-18 |
2020-09-23 |
Merck Patent GmbH |
Matières pour dispositifs électroluminescents organiques
|
WO2015193846A1
(fr)
|
2014-06-20 |
2015-12-23 |
Aurigene Discovery Technologies Limited |
Composés d'imidazole substitués en tant qu'inhibiteurs de l'irak4
|
US11279714B2
(en)
|
2014-06-20 |
2022-03-22 |
Institut Pasteur Korea |
Anti-infective compounds
|
US20170247366A1
(en)
|
2014-06-25 |
2017-08-31 |
Vanderbilt University |
Substituted 4-alkoxypicolinamide analogs as mglur5 negative allosteric modulators and methods of making and using the same
|
KR20160007967A
(ko)
|
2014-07-10 |
2016-01-21 |
삼성디스플레이 주식회사 |
유기 발광 소자
|
WO2016040181A1
(fr)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
3-1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine et ses utilisations thérapeutiques
|
WO2016040180A1
(fr)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
3-1h-benzo[d]imidazol-2-yl)-1h-pyrazolo[3,4-c]pyridine et ses utilisations thérapeutiques
|
WO2016040184A1
(fr)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
3-3h-imidazo[4,5-b]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine et ses utilisations thérapeutiques
|
WO2016040188A1
(fr)
|
2014-09-08 |
2016-03-17 |
Samumed, Llc |
3-3h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-c]pyridine et ses utilisations thérapeutiques
|
WO2016041618A1
(fr)
|
2014-09-15 |
2016-03-24 |
Merck Patent Gmbh |
Indazoles substitués et hétérocycles associés
|
AR102177A1
(es)
|
2014-10-06 |
2017-02-08 |
Merck Patent Gmbh |
Compuestos de heteroarilo como inhibidores de btk y usos de los mismos
|
JO3705B1
(ar)
|
2014-11-26 |
2021-01-31 |
Bayer Pharma AG |
إندازولات مستبدلة جديدة، عمليات لتحضيرها، مستحضرات دوائية تحتوي عليها واستخدامها في إنتاج أدوية
|
CN107206088A
(zh)
|
2014-12-05 |
2017-09-26 |
豪夫迈·罗氏有限公司 |
使用pd‑1轴拮抗剂和hpk1拮抗剂用于治疗癌症的方法和组合物
|
KR102554987B1
(ko)
|
2015-02-03 |
2023-07-12 |
메르크 파텐트 게엠베하 |
금속 착물
|
CN107624110B
(zh)
|
2015-03-06 |
2021-01-26 |
法玛克亚公司 |
赖氨酰氧化酶样2抑制剂及其用途
|
CN112679467B
(zh)
|
2015-03-11 |
2024-11-01 |
Fmc公司 |
杂环取代的二环唑杀有害生物剂
|
WO2016161571A1
(fr)
|
2015-04-08 |
2016-10-13 |
Merck Sharp & Dohme Corp. |
Inhibiteurs de la btk de type indazole et azaindazole
|
CN107872977B
(zh)
|
2015-04-30 |
2021-07-09 |
拜耳制药股份公司 |
Irak4抑制剂与btk抑制剂的组合产品
|
EP3322711B1
(fr)
|
2015-06-25 |
2021-03-10 |
University Health Network |
Inhibiteurs de hpk1 et leurs procédés d'utilisation
|
EP3322409A4
(fr)
|
2015-07-15 |
2019-07-24 |
Aurigene Discovery Technologies Limited |
Composés aza substitués comme inhibiteurs de l'irak-4
|
EP3322698A4
(fr)
|
2015-07-15 |
2019-01-09 |
Aurigene Discovery Technologies Limited |
Composés d'indazole et d'azaindazole à titre d'inhibiteurs d'irak-4
|
EP3331530A4
(fr)
|
2015-08-03 |
2018-12-19 |
Raze Therapeutics Inc. |
Inhibiteurs de mthfd2 et utilisation desdits inhibiteurs
|
WO2017023972A1
(fr)
|
2015-08-03 |
2017-02-09 |
Samumed, Llc. |
3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[4,3-b]pyridines et leurs utilisations thérapeutiques
|
DK3331525T3
(da)
|
2015-08-07 |
2020-12-14 |
Calcimedica Inc |
Anvendelse af CRAC-kanal-inhibitorer til behandling af slagtilfælde og traumatisk hjerneskade
|
WO2017045955A1
(fr)
|
2015-09-14 |
2017-03-23 |
Basf Se |
Composés hétérobicycliques
|
WO2017058915A1
(fr)
|
2015-09-28 |
2017-04-06 |
Araxes Pharma Llc |
Inhibiteurs de protéines mutantes kras g12c
|
WO2017108744A1
(fr)
|
2015-12-22 |
2017-06-29 |
Bayer Pharma Aktiengesellschaft |
Nouveaux indazoles substitués, leurs procédés de préparation, préparations pharmaceutiques les contenant, et leur utilisation pour produire des médicaments
|
US10280164B2
(en)
|
2016-09-09 |
2019-05-07 |
Incyte Corporation |
Pyrazolopyridone compounds and uses thereof
|
CN115819417A
(zh)
|
2016-09-09 |
2023-03-21 |
因赛特公司 |
作为hpk1调节剂的吡唑并吡啶衍生物及其用于治疗癌症的用途
|
WO2018049214A1
(fr)
|
2016-09-09 |
2018-03-15 |
Incyte Corporation |
Dérivés de pyrazolopyridine comme modulateurs de hpk1 et leurs utilisations pour le traitement du cancer
|
TW201811799A
(zh)
|
2016-09-09 |
2018-04-01 |
美商英塞特公司 |
吡唑并嘧啶化合物及其用途
|
US20180228786A1
(en)
|
2017-02-15 |
2018-08-16 |
Incyte Corporation |
Pyrazolopyridine compounds and uses thereof
|
WO2019051199A1
(fr)
|
2017-09-08 |
2019-03-14 |
Incyte Corporation |
Composés de 6-cyano-indazole utilisés en tant que modulateurs de kinase 1 progénitrices hématopoïétiques (hpk1)
|
SG11202007917VA
(en)
|
2018-02-20 |
2020-09-29 |
Incyte Corp |
N-(phenyl)-2-(phenyl)pyrimidine-4-carboxamide derivatives and related compounds as hpk1 inhibitors for treating cancer
|
US10745388B2
(en)
|
2018-02-20 |
2020-08-18 |
Incyte Corporation |
Indazole compounds and uses thereof
|
WO2019164847A1
(fr)
|
2018-02-20 |
2019-08-29 |
Incyte Corporation |
Composés d'indazole et leurs utilisations
|
US11299473B2
(en)
|
2018-04-13 |
2022-04-12 |
Incyte Corporation |
Benzimidazole and indole compounds and uses thereof
|
BR112020021689B1
(pt)
|
2018-04-26 |
2023-02-28 |
Pfizer Inc |
Composto, composição farmacêutica e uso de um composto
|
MA52483A
(fr)
|
2018-05-04 |
2021-03-10 |
Novo Nordisk As |
Dérivés de gip et leurs utilisations
|
MA52623A
(fr)
|
2018-05-17 |
2021-03-24 |
Bayer Ag |
Dérivés de dihydropyrazolo pyrazine carboxamide substitués
|
US10899755B2
(en)
|
2018-08-08 |
2021-01-26 |
Incyte Corporation |
Benzothiazole compounds and uses thereof
|
JP2022543155A
(ja)
|
2019-08-06 |
2022-10-07 |
インサイト・コーポレイション |
Hpk1阻害剤の固体形態
|