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WO2009057569A1 - Préparation pelliculée - Google Patents

Préparation pelliculée Download PDF

Info

Publication number
WO2009057569A1
WO2009057569A1 PCT/JP2008/069487 JP2008069487W WO2009057569A1 WO 2009057569 A1 WO2009057569 A1 WO 2009057569A1 JP 2008069487 W JP2008069487 W JP 2008069487W WO 2009057569 A1 WO2009057569 A1 WO 2009057569A1
Authority
WO
WIPO (PCT)
Prior art keywords
film
coated preparation
disclosed
coated
preparation
Prior art date
Application number
PCT/JP2008/069487
Other languages
English (en)
Japanese (ja)
Inventor
Takeshi Hamaura
Susumu Hasegawa
Ikumasa Ohno
Original Assignee
Daiichi Sankyo Company, Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Sankyo Company, Limited filed Critical Daiichi Sankyo Company, Limited
Priority to CN200880114044A priority Critical patent/CN101842096A/zh
Priority to JP2009539054A priority patent/JPWO2009057569A1/ja
Publication of WO2009057569A1 publication Critical patent/WO2009057569A1/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41781,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/28Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A61K9/2806Coating materials
    • A61K9/2833Organic macromolecular compounds
    • A61K9/284Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/12Drugs for disorders of the urinary system of the kidneys
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/04Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/06Antiarrhythmics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • A61K9/2018Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Hospice & Palliative Care (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

La présente invention concerne une préparation pelliculée, dans laquelle l'odeur de l'agent médicinal qu'elle contient peut être réduite. L'invention concerne spécifiquement une préparation pelliculée qui contient de l'olmésartan médoxomil dans sa formulation, et qui contient de l'alcool polyvinylique ou un copolymère contenant de l'alcool vinylique dans sa pellicule.
PCT/JP2008/069487 2007-10-29 2008-10-28 Préparation pelliculée WO2009057569A1 (fr)

Priority Applications (2)

Application Number Priority Date Filing Date Title
CN200880114044A CN101842096A (zh) 2007-10-29 2008-10-28 薄膜包衣制剂
JP2009539054A JPWO2009057569A1 (ja) 2007-10-29 2008-10-28 フィルムコーティング製剤

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2007280843 2007-10-29
JP2007-280843 2007-10-29

Publications (1)

Publication Number Publication Date
WO2009057569A1 true WO2009057569A1 (fr) 2009-05-07

Family

ID=40590960

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/JP2008/069487 WO2009057569A1 (fr) 2007-10-29 2008-10-28 Préparation pelliculée

Country Status (5)

Country Link
JP (1) JPWO2009057569A1 (fr)
KR (1) KR20100072317A (fr)
CN (1) CN101842096A (fr)
TW (1) TW200927197A (fr)
WO (1) WO2009057569A1 (fr)

Cited By (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011025035A1 (fr) * 2009-08-31 2011-03-03 日新化成株式会社 Composition de revêtement
JP2012193175A (ja) * 2011-03-02 2012-10-11 Daiichi Sankyo Healthcare Co Ltd 速溶性防湿フィルムコーティング製剤及びその製造方法
EP2594277A1 (fr) * 2010-07-07 2013-05-22 Japan Tobacco, Inc. Comprimé contenant du citrate ferrique
WO2014080365A1 (fr) * 2012-11-23 2014-05-30 Ranbaxy Laboratories Limited Procédé de réduction d'une odeur désagréable d'une composition pharmaceutique
WO2014188728A1 (fr) * 2013-05-24 2014-11-27 持田製薬株式会社 Composition pour enrobage par film
EP2830618A4 (fr) * 2012-03-30 2015-08-05 Dae Woong Pharma Composition pharmaceutique comprenant de l'olmésartan médoxomil et de la rosuvastatine ou son sel
JP2016141630A (ja) * 2015-01-30 2016-08-08 富士フイルム株式会社 口腔内崩壊錠
JP2017001999A (ja) * 2015-06-12 2017-01-05 富士フイルム株式会社 薬物含有粒子の製造方法、薬物含有粒子、医薬組成物、及び口腔内崩壊錠
WO2017164208A1 (fr) * 2016-03-24 2017-09-28 第一三共株式会社 Médicament pour le traitement d'une maladie rénale

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102716100B (zh) * 2012-07-12 2013-08-07 南京正大天晴制药有限公司 一种含奥美沙坦酯的片剂及其制备方法

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002179741A (ja) * 2000-10-04 2002-06-26 Basf Ag ヒドロキシアルキル(メタ)アクリレートの水溶性または水分散性(コ)ポリマー、その製造方法、ならびに医薬投与剤形における被覆剤、結合剤および/またはフィルム形成性賦形剤としてのその使用
WO2005019286A1 (fr) * 2003-08-20 2005-03-03 Shionogi & Co., Ltd. Nouvelle composition pour revetements
WO2006123765A1 (fr) * 2005-05-20 2006-11-23 Daiichi Sankyo Company, Limited Preparation recouverte d’un film
WO2006123766A1 (fr) * 2005-05-20 2006-11-23 Daichi Sankyo Company, Limited Preparation recouverte d’un film contenant du dextrose
JP2007091620A (ja) * 2005-09-28 2007-04-12 Kyoto Pharmaceutical Industries Ltd フィルムコーティング錠剤
JP2007197410A (ja) * 2006-01-30 2007-08-09 Lion Corp フィルムコーティング錠

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2002179741A (ja) * 2000-10-04 2002-06-26 Basf Ag ヒドロキシアルキル(メタ)アクリレートの水溶性または水分散性(コ)ポリマー、その製造方法、ならびに医薬投与剤形における被覆剤、結合剤および/またはフィルム形成性賦形剤としてのその使用
WO2005019286A1 (fr) * 2003-08-20 2005-03-03 Shionogi & Co., Ltd. Nouvelle composition pour revetements
WO2006123765A1 (fr) * 2005-05-20 2006-11-23 Daiichi Sankyo Company, Limited Preparation recouverte d’un film
WO2006123766A1 (fr) * 2005-05-20 2006-11-23 Daichi Sankyo Company, Limited Preparation recouverte d’un film contenant du dextrose
JP2007091620A (ja) * 2005-09-28 2007-04-12 Kyoto Pharmaceutical Industries Ltd フィルムコーティング錠剤
JP2007197410A (ja) * 2006-01-30 2007-08-09 Lion Corp フィルムコーティング錠

Cited By (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011025035A1 (fr) * 2009-08-31 2011-03-03 日新化成株式会社 Composition de revêtement
JP5730205B2 (ja) * 2009-08-31 2015-06-03 日新化成株式会社 コーティング用組成物
EP2594277A1 (fr) * 2010-07-07 2013-05-22 Japan Tobacco, Inc. Comprimé contenant du citrate ferrique
EP2594277A4 (fr) * 2010-07-07 2014-01-01 Japan Tobacco Inc Comprimé contenant du citrate ferrique
JP2012193175A (ja) * 2011-03-02 2012-10-11 Daiichi Sankyo Healthcare Co Ltd 速溶性防湿フィルムコーティング製剤及びその製造方法
EP2830618A4 (fr) * 2012-03-30 2015-08-05 Dae Woong Pharma Composition pharmaceutique comprenant de l'olmésartan médoxomil et de la rosuvastatine ou son sel
WO2014080365A1 (fr) * 2012-11-23 2014-05-30 Ranbaxy Laboratories Limited Procédé de réduction d'une odeur désagréable d'une composition pharmaceutique
WO2014188728A1 (fr) * 2013-05-24 2014-11-27 持田製薬株式会社 Composition pour enrobage par film
JPWO2014188728A1 (ja) * 2013-05-24 2017-02-23 持田製薬株式会社 フィルムコーティング用組成物
JP2016141630A (ja) * 2015-01-30 2016-08-08 富士フイルム株式会社 口腔内崩壊錠
JP2017001999A (ja) * 2015-06-12 2017-01-05 富士フイルム株式会社 薬物含有粒子の製造方法、薬物含有粒子、医薬組成物、及び口腔内崩壊錠
WO2017164208A1 (fr) * 2016-03-24 2017-09-28 第一三共株式会社 Médicament pour le traitement d'une maladie rénale

Also Published As

Publication number Publication date
CN101842096A (zh) 2010-09-22
JPWO2009057569A1 (ja) 2011-03-10
TW200927197A (en) 2009-07-01
KR20100072317A (ko) 2010-06-30

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