WO2008147169A8 - Microémulsion contenant de la pirfénidone - Google Patents
Microémulsion contenant de la pirfénidone Download PDFInfo
- Publication number
- WO2008147169A8 WO2008147169A8 PCT/MX2008/000068 MX2008000068W WO2008147169A8 WO 2008147169 A8 WO2008147169 A8 WO 2008147169A8 MX 2008000068 W MX2008000068 W MX 2008000068W WO 2008147169 A8 WO2008147169 A8 WO 2008147169A8
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- microemulsion containing
- containing pirfenidone
- pirfenidone
- microemulsion
- capsules
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4412—Non condensed pyridines; Hydrogenated derivatives thereof having oxo groups directly attached to the heterocyclic ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0087—Galenical forms not covered by A61K9/02 - A61K9/7023
- A61K9/0095—Drinks; Beverages; Syrups; Compositions for reconstitution thereof, e.g. powders or tablets to be dispersed in a glass of water; Veterinary drenches
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/107—Emulsions ; Emulsion preconcentrates; Micelles
- A61K9/1075—Microemulsions or submicron emulsions; Preconcentrates or solids thereof; Micelles, e.g. made of phospholipids or block copolymers
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Biophysics (AREA)
- Molecular Biology (AREA)
- Dispersion Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Abstract
La présente invention concerne une composition microémulsionnable de Pirfénidone, qui présente des avantages par rapport à d'autres formes pharmaceutiques à administrer par voie orale connues dans l'état de la technique, comme des comprimés, capsules, suspensions et solutions.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
MX2007006438 | 2007-05-29 | ||
MXMX/A/2007/006348 | 2007-05-29 |
Publications (3)
Publication Number | Publication Date |
---|---|
WO2008147169A2 WO2008147169A2 (fr) | 2008-12-04 |
WO2008147169A3 WO2008147169A3 (fr) | 2009-01-22 |
WO2008147169A8 true WO2008147169A8 (fr) | 2009-07-30 |
Family
ID=40075678
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/MX2008/000068 WO2008147169A2 (fr) | 2007-05-29 | 2008-05-29 | Microémulsion contenant de la pirfénidone |
Country Status (1)
Country | Link |
---|---|
WO (1) | WO2008147169A2 (fr) |
Families Citing this family (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2296653B1 (fr) | 2008-06-03 | 2016-01-27 | Intermune, Inc. | Composés et procédés de traitement des troubles inflammatoires et fibrotiques |
CN102846555B (zh) * | 2012-04-09 | 2014-06-25 | 珠海亿邦制药股份有限公司 | 一种以吡非尼酮为活性成分的固体制剂及其应用 |
AR092742A1 (es) | 2012-10-02 | 2015-04-29 | Intermune Inc | Piridinonas antifibroticas |
CN110452216B (zh) | 2014-04-02 | 2022-08-26 | 英特穆恩公司 | 抗纤维化吡啶酮类 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1113798B1 (fr) * | 1998-09-18 | 2003-01-02 | Mepha AG | Formulation topique a base d'alkyl-, phenyl-pyridone |
CH696420A5 (de) * | 2002-09-13 | 2007-06-15 | Mepha Ag | Neue stabile Zubereitungen von Alkyl-, Phenyl-Pyridonen für topische Anwendung. |
JP4542743B2 (ja) * | 2002-12-26 | 2010-09-15 | Kdl株式会社 | ピリドン誘導体の溶液状医薬組成物 |
NZ591443A (en) * | 2005-09-22 | 2013-04-26 | Intermune Inc | Granule formation of pirfenidone and pharmaceutically acceptable excipients |
-
2008
- 2008-05-29 WO PCT/MX2008/000068 patent/WO2008147169A2/fr active Application Filing
Also Published As
Publication number | Publication date |
---|---|
WO2008147169A2 (fr) | 2008-12-04 |
WO2008147169A3 (fr) | 2009-01-22 |
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