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WO2008065527A3 - Gallic acid esters of fragrant alcohols - Google Patents

Gallic acid esters of fragrant alcohols Download PDF

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Publication number
WO2008065527A3
WO2008065527A3 PCT/IB2007/003804 IB2007003804W WO2008065527A3 WO 2008065527 A3 WO2008065527 A3 WO 2008065527A3 IB 2007003804 W IB2007003804 W IB 2007003804W WO 2008065527 A3 WO2008065527 A3 WO 2008065527A3
Authority
WO
WIPO (PCT)
Prior art keywords
gallic acid
acid esters
fragrant alcohols
fragrant
alcohols
Prior art date
Application number
PCT/IB2007/003804
Other languages
French (fr)
Other versions
WO2008065527A2 (en
Inventor
Carlo Ghisalberti
Original Assignee
Carlo Ghisalberti
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from ITMI20062269 external-priority patent/ITMI20062269A1/en
Priority claimed from ITMI20062317 external-priority patent/ITMI20062317A1/en
Priority claimed from ITMI20062351 external-priority patent/ITMI20062351A1/en
Priority claimed from ITMI20062350 external-priority patent/ITMI20062350A1/en
Application filed by Carlo Ghisalberti filed Critical Carlo Ghisalberti
Publication of WO2008065527A2 publication Critical patent/WO2008065527A2/en
Publication of WO2008065527A3 publication Critical patent/WO2008065527A3/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
    • C07C69/76—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring
    • C07C69/84—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring
    • C07C69/88—Esters of carboxylic acids having a carboxyl group bound to a carbon atom of a six-membered aromatic ring of monocyclic hydroxy carboxylic acids, the hydroxy groups and the carboxyl groups of which are bound to carbon atoms of a six-membered aromatic ring with esterified carboxyl groups
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/33—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing oxygen
    • A61K8/37—Esters of carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00—Cosmetics or similar toiletry preparations
    • A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
    • A61K8/4973—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with oxygen as the only hetero atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/10—Anti-acne agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/14—Drugs for dermatological disorders for baldness or alopecia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00—Preparations for care of the skin
    • A61Q19/008—Preparations for oily skin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/74—Biological properties of particular ingredients
    • A61K2800/78—Enzyme modulators, e.g. Enzyme agonists
    • A61K2800/782—Enzyme inhibitors; Enzyme antagonists
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/14—The ring being saturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00—Systems containing only non-condensed rings
    • C07C2601/12—Systems containing only non-condensed rings with a six-membered ring
    • C07C2601/16—Systems containing only non-condensed rings with a six-membered ring the ring being unsaturated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2602/00—Systems containing two condensed rings
    • C07C2602/36—Systems containing two condensed rings the rings having more than two atoms in common
    • C07C2602/42—Systems containing two condensed rings the rings having more than two atoms in common the bicyclo ring system containing seven carbon atoms

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Dermatology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Birds (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

Gallates formed by condensation of gallic acid with a hydroxyl-containing fragrance for the use in a composition suitable for disinfecting and seboregulating purposes.
PCT/IB2007/003804 2006-11-27 2007-12-06 Gallic acid esters of fragrant alcohols WO2008065527A2 (en)

Applications Claiming Priority (8)

Application Number Priority Date Filing Date Title
ITMI2006A002269 2006-11-27
ITMI20062269 ITMI20062269A1 (en) 2006-11-27 2006-11-27 OMEGA-INSATURAL ESTERS OF GALLIC ACID AND THEIR APPLICATIONS
ITMI2006A002317 2006-12-01
ITMI20062317 ITMI20062317A1 (en) 2006-12-01 2006-12-01 INSATURAL ESTERS OF GALLIC ACID
ITMI20062351 ITMI20062351A1 (en) 2006-12-06 2006-12-06 PHENOLIC ESTERS OF GALLIC ACID IN THE TREATMENT OF ANDROGENETIC DISORDERS
ITMI20062350 ITMI20062350A1 (en) 2006-12-06 2006-12-06 TERPENIC ESTERS OF GALLIC ACID IN THE TREATMENT OF ANDROGENETIC DISORDERS
ITMI2006A002351 2006-12-06
ITMI2006A002350 2006-12-06

Publications (2)

Publication Number Publication Date
WO2008065527A2 WO2008065527A2 (en) 2008-06-05
WO2008065527A3 true WO2008065527A3 (en) 2008-08-07

Family

ID=39306458

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/IB2007/003804 WO2008065527A2 (en) 2006-11-27 2007-12-06 Gallic acid esters of fragrant alcohols

Country Status (1)

Country Link
WO (1) WO2008065527A2 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011138345A2 (en) 2010-05-06 2011-11-10 Basf Se Fungicidal mixtures based on gallic acid esters
MX365561B (en) 2012-12-27 2019-06-05 Kimberly Clark Co Water soluble essential oils and their use.
WO2014101051A1 (en) * 2012-12-27 2014-07-03 Kimberly-Clark Worldwide, Inc. Water soluble farnesol analogs and their use
CN114315587B (en) * 2021-12-23 2023-12-08 江苏浩丰生物科技有限公司 Linalyl vanillate, preparation method thereof and application thereof in tobacco industry
CN115124425B (en) * 2022-06-27 2023-10-17 浙江海昇药业股份有限公司 3, 5-dibromo-4-hydroxybenzoic acid dimer, synthesis method and application thereof

Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4394389A (en) * 1979-03-01 1983-07-19 Riet Bartholomeus Van T Hydroxybenzohydroxamic acids, benzamides and esters as ribonucleotide reductase inhibitors
WO1999022728A1 (en) * 1997-10-31 1999-05-14 Arch Development Corporation Methods and compositions for regulation of 5-alpha reductase activity
WO2004073707A1 (en) * 2003-02-19 2004-09-02 Unilever N.V. Topical composition containing alkyl gallate or alkyl hydroxybenzoate or phenol alkyloxy as agent against acne
JP2005281164A (en) * 2004-03-29 2005-10-13 Api Co Ltd Gallic ester compound, method for producing the same, anticancer agent and preparation
EP1604660A1 (en) * 2003-01-29 2005-12-14 Alps Pharmaceutical Ind. Co. Ltd. Medicinal composition for treating infection with drug-resistant staphylococcus aureus

Patent Citations (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4394389A (en) * 1979-03-01 1983-07-19 Riet Bartholomeus Van T Hydroxybenzohydroxamic acids, benzamides and esters as ribonucleotide reductase inhibitors
WO1999022728A1 (en) * 1997-10-31 1999-05-14 Arch Development Corporation Methods and compositions for regulation of 5-alpha reductase activity
EP1604660A1 (en) * 2003-01-29 2005-12-14 Alps Pharmaceutical Ind. Co. Ltd. Medicinal composition for treating infection with drug-resistant staphylococcus aureus
WO2004073707A1 (en) * 2003-02-19 2004-09-02 Unilever N.V. Topical composition containing alkyl gallate or alkyl hydroxybenzoate or phenol alkyloxy as agent against acne
JP2005281164A (en) * 2004-03-29 2005-10-13 Api Co Ltd Gallic ester compound, method for producing the same, anticancer agent and preparation

Non-Patent Citations (7)

* Cited by examiner, † Cited by third party
Title
DATABASE CA [online] CHEMICAL ABSTRACTS SERVICE, COLUMBUS, OHIO, US; TAZAWA, SHIGEMI ET AL: "Enzymic preparation of gallic acid esters as anticancer agents", XP002481674, retrieved from STN Database accession no. 2005:1102569 *
HAK HEE KANG ET AL: "DEPIGMENTING ACTIVITY AND LOW CYTOTOXICITY OF ALKOXY BENZOATES OR ALKOXY CINNAMTE IN CULTURED MELANOCYTES", CHEMICAL AND PHARMACEUTICAL BULLETIN, PHARMACEUTICAL SOCIETY OF JAPAN, TOKYO, vol. 51, no. 9, 1 September 2003 (2003-09-01), pages 1085 - 1088, XP008054792, ISSN: 0009-2363 *
IKURO ABE, YASUHIKO KASHIWAGI AND HIROSHI NOGUCHI: "Inhibition of vertebrate squalene epoxidase by isoprenyl gallates and phenylalkyl gallates", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 10, no. 22, 20 November 2000 (2000-11-20), GBOXFORD, pages 2525 - 2528, XP002481672 *
ISAO KUBO, KEN-ICHI FUJITA, KEN-ICHI NIHEI: "Molecular design of multifunctional antibacterial agents against methicillin resistant Staphylococcus aureus (MRSA)", BIOORGANIC & MEDICINAL CHEMISTRY., vol. 11, 2003, GBELSEVIER SCIENCE LTD., pages 4255 - 4262, XP002481670 *
ISAO KUBO,* PING XIAO, KEN-ICHI NIHEI, KEN-ICHI FUJITA, YOSHIRO YAMAGIWA, AND TADAO KAMIKAWA: "Molecular Design of Antifungal Agents", JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY., vol. 50, 2002, USAMERICAN CHEMICAL SOCIETY. WASHINGTON., pages 3992 - 3998, XP002481671 *
L. M. VIRANGA TILLEKERATNE, ANGELA SHERETTE, JENNIFER A. FULMER, LYNN HUPE, DONALD HUPE, SAM GABBARA ET AL.: "Differential Inhibition of polymerase and Strand-Transfer Activities of HIV-1 Reverse Transcriptase", BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, vol. 12, no. 4, 2002, GBOXFORD, pages 525 - 528, XP002481673 *
NAKAMURA E S ET AL: "Cancer chemopreventive effects of constituents of Caesalpinia ferrea and related compounds", CANCER LETTERS, NEW YORK, NY, US, vol. 177, no. 2, 1 January 2002 (2002-01-01), pages 119 - 124, XP002996965, ISSN: 0304-3835 *

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Publication number Publication date
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