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WO2007048223A3 - Systeme d'administration de medicaments a retention gastrique - Google Patents

Systeme d'administration de medicaments a retention gastrique Download PDF

Info

Publication number
WO2007048223A3
WO2007048223A3 PCT/CA2006/001706 CA2006001706W WO2007048223A3 WO 2007048223 A3 WO2007048223 A3 WO 2007048223A3 CA 2006001706 W CA2006001706 W CA 2006001706W WO 2007048223 A3 WO2007048223 A3 WO 2007048223A3
Authority
WO
WIPO (PCT)
Prior art keywords
delivery system
drug delivery
gastric retention
matrix component
intermingled
Prior art date
Application number
PCT/CA2006/001706
Other languages
English (en)
Other versions
WO2007048223A2 (fr
Inventor
Jack Aurora
Vinayak Sant
Original Assignee
Pharmascience Inc
Jack Aurora
Vinayak Sant
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from CA 2524422 external-priority patent/CA2524422A1/fr
Priority claimed from US11/257,361 external-priority patent/US20070092565A1/en
Application filed by Pharmascience Inc, Jack Aurora, Vinayak Sant filed Critical Pharmascience Inc
Priority to EP06804634A priority Critical patent/EP1957052A2/fr
Publication of WO2007048223A2 publication Critical patent/WO2007048223A2/fr
Publication of WO2007048223A3 publication Critical patent/WO2007048223A3/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/30Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
    • A61K47/36Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
    • A61K47/38Cellulose; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0065Forms with gastric retention, e.g. floating on gastric juice, adhering to gastric mucosa, expanding to prevent passage through the pylorus

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Medicinal Preparation (AREA)

Abstract

L'invention concerne un système d'administration de médicaments à rétention gastrique (c.-à-d. une forme pharmaceutique à libération contrôlée) formulé pour favoriser la rétention de la forme pharmaceutique dans le tractus gastro-intestinal supérieur et en particulier dans l'estomac.
PCT/CA2006/001706 2005-10-25 2006-10-17 Systeme d'administration de medicaments a retention gastrique WO2007048223A2 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
EP06804634A EP1957052A2 (fr) 2005-10-25 2006-10-17 Systeme d'administration de medicaments a retention gastrique

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CA 2524422 CA2524422A1 (fr) 2005-10-25 2005-10-25 Dispositif d'administration de medicament a retention gastrique
US11/257,361 2005-10-25
CA2,524,422 2005-10-25
US11/257,361 US20070092565A1 (en) 2005-10-25 2005-10-25 Gastric retention drug delivery system

Publications (2)

Publication Number Publication Date
WO2007048223A2 WO2007048223A2 (fr) 2007-05-03
WO2007048223A3 true WO2007048223A3 (fr) 2007-06-14

Family

ID=37968169

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/CA2006/001706 WO2007048223A2 (fr) 2005-10-25 2006-10-17 Systeme d'administration de medicaments a retention gastrique

Country Status (2)

Country Link
EP (1) EP1957052A2 (fr)
WO (1) WO2007048223A2 (fr)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2010143052A1 (fr) * 2009-06-12 2010-12-16 Micro Labs Limited Nouvelles compositions pharmaceutiques contenant de la prégabaline
EP2361615A1 (fr) 2010-02-19 2011-08-31 Alfred E. Tiefenbacher GmbH & Co. KG Comprimé à libération prolongée de dipyridamole
MX2012013021A (es) * 2010-05-11 2012-12-17 Cima Labs Inc Formulaciones resistentes a alcohol.
EP2415460A1 (fr) * 2010-08-03 2012-02-08 ratiopharm GmbH Formulations pour l'administration orale de prégabaline
WO2013109199A1 (fr) * 2011-12-19 2013-07-25 Mahmut Bilgic Formulations pharmaceutiques effervescentes comprenant de la prégabaline et de la vitamine b12
WO2013100874A1 (fr) * 2011-12-19 2013-07-04 Mahmut Bilgic Formulation de prégabline effervescente
EP2698144A1 (fr) * 2012-08-12 2014-02-19 Ali Raif Ilaç Sanayi ve Ticaret Anonim Sirketi Formulation de comprimé à libération prolongée contenant de la gabapentine dont l'aptitude à rester dans l'estomac est améliorée
WO2015114509A1 (fr) * 2014-01-28 2015-08-06 Ranbaxy Laboratories Limited Comprimés à rétention gastrique stabilisée de prégabaline
CA2951909C (fr) 2014-06-11 2022-08-16 Massachusetts Institute Of Technology Dispositifs a demeure auto-assembles, et procedes associes
US20170266112A1 (en) 2014-06-11 2017-09-21 Massachusetts Institute Of Technology Residence structures and related methods
CN107592803B (zh) 2015-05-01 2021-01-22 麻省理工学院 可触发形状记忆感应装置
EP3364946A4 (fr) 2015-10-23 2019-06-26 Lyndra, Inc. Systèmes à demeure gastriques pour libération prolongée d'agents thérapeutiques et leurs procédés d'utilisation
JP7030052B2 (ja) 2015-12-08 2022-03-04 リンドラ セラピューティクス, インコーポレイティド 胃滞留システムのための幾何学的構成
CN109310639A (zh) 2016-05-27 2019-02-05 林德拉有限公司 用于胃驻留系统的材料结构
EP3518902A4 (fr) 2016-09-30 2020-07-08 Lyndra, Inc. Systèmes de résidence gastrique permettant l'administration prolongée de médicaments de la classe de l'adamantane
US12023406B2 (en) 2017-06-09 2024-07-02 Lyndra Therapeutics, Inc. Gastric residence systems with release rate-modulating films
CN113521023B (zh) * 2021-07-16 2023-04-25 昆明理工大学 一种紫胶树脂基胃内漂浮滞留载药系统的制备方法

Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0941064A1 (fr) * 1996-11-17 1999-09-15 Yissum Research Development Company Of The Hebrew University Of Jerusalem PREPARATIONS PHARMACEUTIQUES SERVANT A EFFECTUER LA LIBERATION CONTROLEE D'ANTIBIOTIQUES DE beta-LACTAME
CA2452738A1 (fr) * 2001-07-04 2003-02-13 Sun Pharmaceutical Industries Limited Systeme d'administration regulee de medicament a retention gastrique
WO2003026637A2 (fr) * 2001-09-28 2003-04-03 Sun Pharmaceutical Industries Limited Forme posologique pour traiter le diabete sucre
WO2004032906A1 (fr) * 2002-10-11 2004-04-22 Depomed Development, Ltd. Forme gastro-retentive pour administrer du levodopa
US6861072B1 (en) * 1998-10-16 2005-03-01 Sanofi-Synthelabo Pharmaceutical composition with gastric residence and controlled release
WO2005060942A1 (fr) * 2003-12-19 2005-07-07 Aurobindo Pharma Ltd Composition pharmaceutique de metformine a liberation prolongee
US20060159743A1 (en) * 2001-10-25 2006-07-20 Depomed, Inc. Methods of treating non-nociceptive pain states with gastric retentive gabapentin
US20060165745A1 (en) * 2005-01-21 2006-07-27 Yiwen Chew Sustained release tablets for treatment of aqueous environment and methods for making the same

Patent Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0941064A1 (fr) * 1996-11-17 1999-09-15 Yissum Research Development Company Of The Hebrew University Of Jerusalem PREPARATIONS PHARMACEUTIQUES SERVANT A EFFECTUER LA LIBERATION CONTROLEE D'ANTIBIOTIQUES DE beta-LACTAME
US6861072B1 (en) * 1998-10-16 2005-03-01 Sanofi-Synthelabo Pharmaceutical composition with gastric residence and controlled release
CA2452738A1 (fr) * 2001-07-04 2003-02-13 Sun Pharmaceutical Industries Limited Systeme d'administration regulee de medicament a retention gastrique
WO2003026637A2 (fr) * 2001-09-28 2003-04-03 Sun Pharmaceutical Industries Limited Forme posologique pour traiter le diabete sucre
US20060159743A1 (en) * 2001-10-25 2006-07-20 Depomed, Inc. Methods of treating non-nociceptive pain states with gastric retentive gabapentin
WO2004032906A1 (fr) * 2002-10-11 2004-04-22 Depomed Development, Ltd. Forme gastro-retentive pour administrer du levodopa
WO2005060942A1 (fr) * 2003-12-19 2005-07-07 Aurobindo Pharma Ltd Composition pharmaceutique de metformine a liberation prolongee
US20060165745A1 (en) * 2005-01-21 2006-07-27 Yiwen Chew Sustained release tablets for treatment of aqueous environment and methods for making the same

Also Published As

Publication number Publication date
EP1957052A2 (fr) 2008-08-20
WO2007048223A2 (fr) 2007-05-03

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