WO2003011859A3 - Derives oxazolidinones utilises en tant qu'agents antibacteriens - Google Patents
Derives oxazolidinones utilises en tant qu'agents antibacteriens Download PDFInfo
- Publication number
- WO2003011859A3 WO2003011859A3 PCT/GB2002/003404 GB0203404W WO03011859A3 WO 2003011859 A3 WO2003011859 A3 WO 2003011859A3 GB 0203404 W GB0203404 W GB 0203404W WO 03011859 A3 WO03011859 A3 WO 03011859A3
- Authority
- WO
- WIPO (PCT)
- Prior art keywords
- alkyl
- antibacterial agents
- substituted
- oxazolidinone derivatives
- group
- Prior art date
Links
- IZXIZTKNFFYFOF-UHFFFAOYSA-N 2-Oxazolidone Chemical class O=C1NCCO1 IZXIZTKNFFYFOF-UHFFFAOYSA-N 0.000 title 1
- 239000003242 anti bacterial agent Substances 0.000 title 1
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 3
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- QGZKDVFQNNGYKY-UHFFFAOYSA-O Ammonium Chemical group [NH4+] QGZKDVFQNNGYKY-UHFFFAOYSA-O 0.000 abstract 1
- 101100294115 Caenorhabditis elegans nhr-4 gene Proteins 0.000 abstract 1
- 229910019142 PO4 Inorganic materials 0.000 abstract 1
- 125000004423 acyloxy group Chemical group 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000001118 alkylidene group Chemical group 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 229910052736 halogen Inorganic materials 0.000 abstract 1
- 150000002367 halogens Chemical group 0.000 abstract 1
- 125000005842 heteroatom Chemical group 0.000 abstract 1
- 125000005462 imide group Chemical group 0.000 abstract 1
- 150000002917 oxazolidines Chemical class 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- NBIIXXVUZAFLBC-UHFFFAOYSA-K phosphate Chemical group [O-]P([O-])([O-])=O NBIIXXVUZAFLBC-UHFFFAOYSA-K 0.000 abstract 1
- 239000010452 phosphate Chemical group 0.000 abstract 1
- 229920006395 saturated elastomer Polymers 0.000 abstract 1
- -1 substituted aryl sulphonate Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB0118407.6 | 2001-07-27 | ||
GBGB0118407.6A GB0118407D0 (en) | 2001-07-27 | 2001-07-27 | Oxazolidinone derivatives as antibacterial agents |
Related Child Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
US10/719,232 Continuation US6908013B2 (en) | 2001-05-25 | 2003-11-20 | Tamper-evident device |
Publications (2)
Publication Number | Publication Date |
---|---|
WO2003011859A2 WO2003011859A2 (fr) | 2003-02-13 |
WO2003011859A3 true WO2003011859A3 (fr) | 2003-04-03 |
Family
ID=9919346
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PCT/GB2002/003404 WO2003011859A2 (fr) | 2001-07-27 | 2002-07-25 | Derives oxazolidinones utilises en tant qu'agents antibacteriens |
Country Status (2)
Country | Link |
---|---|
GB (1) | GB0118407D0 (fr) |
WO (1) | WO2003011859A2 (fr) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
YU52403A (sh) | 2000-12-26 | 2006-03-03 | Dr.Reddy's Research Foundation | Heterociklična jedinjenja koja imaju antibakterijsko dejstvo, postupak za njihovo dobijanje i farmaceutske smeše koje ih sadrže |
US7160912B2 (en) | 2000-12-26 | 2007-01-09 | Dr.Reddy's Laboratories Ltd. | Heterocyclic compounds having antibacterial activity: process for their preparation and pharmaceutical compositions containing them |
US7396847B2 (en) | 2001-09-11 | 2008-07-08 | Astrazeneca Ab | Oxazolidinone and/or isoxazoline as antibacterial agents |
EP2181993A1 (fr) | 2006-03-31 | 2010-05-05 | Research Foundation Itsuu Laboratory | Dérivés d'oxazolidinone antimicrobiens |
US7538107B2 (en) | 2006-08-15 | 2009-05-26 | Wyeth | Oxazinan-2-one derivatives useful as PR modulators |
TW200815428A (en) | 2006-08-15 | 2008-04-01 | Wyeth Corp | Oxazolidone derivatives as PR modulators |
WO2008021338A2 (fr) | 2006-08-15 | 2008-02-21 | Wyeth | Dérivés d'oxazolidone tricycliques utiles en tant que modulateurs du récepteur de la progestérone |
US7649007B2 (en) | 2006-08-15 | 2010-01-19 | Wyeth Llc | Oxazolidine derivatives as PR modulators |
US7652018B2 (en) | 2006-08-15 | 2010-01-26 | Wyeth Llc | Imidazolidin-2-one derivatives useful as PR modulators |
EP2669283A1 (fr) | 2007-10-02 | 2013-12-04 | Shionogi&Co., Ltd. | Dérivé dýoxazolidinone doté dýune bague hétéro composée de 7 éléments |
CN116423599B (zh) * | 2023-05-29 | 2024-06-25 | 德华兔宝宝装饰新材股份有限公司 | 抗菌阻燃木单板及其制备方法 |
Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0359418A1 (fr) * | 1988-09-15 | 1990-03-21 | The Upjohn Company | 5-Indolinyl-5-bêta amidométhyloxazolidines-2-one, 3-(phényl condensé)-5 bêta amidométhyloxazolidines-2-ones et 3-phényl-azoté-5 bêta amidométhyloxazolidine 2-one |
EP0693491A1 (fr) * | 1994-07-20 | 1996-01-24 | Bayer Ag | Oxazolidinones substituées par un groupe hétéroaryle à 5 chaínons comme médicament anti-bactérien |
WO1997021708A1 (fr) * | 1995-12-13 | 1997-06-19 | Pharmacia & Upjohn Company | Derives de 4-pyrimidinyl- ou 4-pyrazinyl-piperazinyl-phenyl-oxazolidinone, leur preparation et leur emploi comme agents antibacteriens |
WO1999002525A1 (fr) * | 1997-07-11 | 1999-01-21 | Pharmacia & Upjohn Company | Agents antibacteriens de type phenyloxazolidinones de thiadiazolyle et d'oxadiazolyle |
-
2001
- 2001-07-27 GB GBGB0118407.6A patent/GB0118407D0/en not_active Ceased
-
2002
- 2002-07-25 WO PCT/GB2002/003404 patent/WO2003011859A2/fr not_active Application Discontinuation
Patent Citations (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP0359418A1 (fr) * | 1988-09-15 | 1990-03-21 | The Upjohn Company | 5-Indolinyl-5-bêta amidométhyloxazolidines-2-one, 3-(phényl condensé)-5 bêta amidométhyloxazolidines-2-ones et 3-phényl-azoté-5 bêta amidométhyloxazolidine 2-one |
EP0693491A1 (fr) * | 1994-07-20 | 1996-01-24 | Bayer Ag | Oxazolidinones substituées par un groupe hétéroaryle à 5 chaínons comme médicament anti-bactérien |
WO1997021708A1 (fr) * | 1995-12-13 | 1997-06-19 | Pharmacia & Upjohn Company | Derives de 4-pyrimidinyl- ou 4-pyrazinyl-piperazinyl-phenyl-oxazolidinone, leur preparation et leur emploi comme agents antibacteriens |
WO1999002525A1 (fr) * | 1997-07-11 | 1999-01-21 | Pharmacia & Upjohn Company | Agents antibacteriens de type phenyloxazolidinones de thiadiazolyle et d'oxadiazolyle |
Also Published As
Publication number | Publication date |
---|---|
GB0118407D0 (en) | 2001-09-19 |
WO2003011859A2 (fr) | 2003-02-13 |
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