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WO2001028590A3 - COMPOSITIONS PHARMACEUTIQUES RENFERMANT UN ESTER N-[N-(3,3-DIMETHYLBUTYL)-1-α-ASPARTYL]-L-PHENYLALANINE METHYL - Google Patents

COMPOSITIONS PHARMACEUTIQUES RENFERMANT UN ESTER N-[N-(3,3-DIMETHYLBUTYL)-1-α-ASPARTYL]-L-PHENYLALANINE METHYL Download PDF

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Publication number
WO2001028590A3
WO2001028590A3 PCT/US2000/028731 US0028731W WO0128590A3 WO 2001028590 A3 WO2001028590 A3 WO 2001028590A3 US 0028731 W US0028731 W US 0028731W WO 0128590 A3 WO0128590 A3 WO 0128590A3
Authority
WO
WIPO (PCT)
Prior art keywords
aspartyl
dimethylbutyl
pharmaceutical compositions
methyl ester
compositions containing
Prior art date
Application number
PCT/US2000/028731
Other languages
English (en)
Other versions
WO2001028590A2 (fr
Inventor
Subbarao V Ponakala
Original Assignee
Nutrasweet Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nutrasweet Co filed Critical Nutrasweet Co
Priority to AU10934/01A priority Critical patent/AU1093401A/en
Publication of WO2001028590A2 publication Critical patent/WO2001028590A2/fr
Publication of WO2001028590A3 publication Critical patent/WO2001028590A3/fr

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2013Organic compounds, e.g. phospholipids, fats
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23LFOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES, NOT OTHERWISE PROVIDED FOR; PREPARATION OR TREATMENT THEREOF
    • A23L27/00Spices; Flavouring agents or condiments; Artificial sweetening agents; Table salts; Dietetic salt substitutes; Preparation or treatment thereof
    • A23L27/30Artificial sweetening agents
    • A23L27/31Artificial sweetening agents containing amino acids, nucleotides, peptides or derivatives
    • A23L27/32Artificial sweetening agents containing amino acids, nucleotides, peptides or derivatives containing dipeptides or derivatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/06Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
    • A61K47/16Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing nitrogen, e.g. nitro-, nitroso-, azo-compounds, nitriles, cyanates
    • A61K47/18Amines; Amides; Ureas; Quaternary ammonium compounds; Amino acids; Oligopeptides having up to five amino acids
    • A61K47/183Amino acids, e.g. glycine, EDTA or aspartame
    • AHUMAN NECESSITIES
    • A23FOODS OR FOODSTUFFS; TREATMENT THEREOF, NOT COVERED BY OTHER CLASSES
    • A23VINDEXING SCHEME RELATING TO FOODS, FOODSTUFFS OR NON-ALCOHOLIC BEVERAGES AND LACTIC OR PROPIONIC ACID BACTERIA USED IN FOODSTUFFS OR FOOD PREPARATION
    • A23V2002/00Food compositions, function of food ingredients or processes for food or foodstuffs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0053Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Nutrition Science (AREA)
  • Food Science & Technology (AREA)
  • Polymers & Plastics (AREA)
  • Medicinal Preparation (AREA)
  • Seasonings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

L'invention concerne des produits pharmaceutiques et des compositions associées renfermant du néotame. Ces compositions pharmaceutiques ont démontré avoir des caractéristiques de goût et d'arôme améliorées.
PCT/US2000/028731 1999-10-19 2000-10-18 COMPOSITIONS PHARMACEUTIQUES RENFERMANT UN ESTER N-[N-(3,3-DIMETHYLBUTYL)-1-α-ASPARTYL]-L-PHENYLALANINE METHYL WO2001028590A2 (fr)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AU10934/01A AU1093401A (en) 1999-10-19 2000-10-18 Pharmaceutical compositions containing n-(n-(3,3-dimethylbutyl)-1-alpha-aspartyl)-l-phenylalanine methyl ester

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US16030599P 1999-10-19 1999-10-19
US60/160,305 1999-10-19

Publications (2)

Publication Number Publication Date
WO2001028590A2 WO2001028590A2 (fr) 2001-04-26
WO2001028590A3 true WO2001028590A3 (fr) 2008-01-03

Family

ID=22576354

Family Applications (1)

Application Number Title Priority Date Filing Date
PCT/US2000/028731 WO2001028590A2 (fr) 1999-10-19 2000-10-18 COMPOSITIONS PHARMACEUTIQUES RENFERMANT UN ESTER N-[N-(3,3-DIMETHYLBUTYL)-1-α-ASPARTYL]-L-PHENYLALANINE METHYL

Country Status (2)

Country Link
AU (1) AU1093401A (fr)
WO (1) WO2001028590A2 (fr)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2859603B1 (fr) * 2003-09-11 2005-12-30 Christian Fenioux Utilisation de la neohesperidine dihydrochalcone dans des compositions orales comprenant des vitamines et/ou des mineraux
JP5852783B2 (ja) * 2011-02-25 2016-02-03 小川香料株式会社 高甘味度甘味料の呈味改善剤
GB2551987A (en) 2016-07-01 2018-01-10 Gw Res Ltd Oral cannabinoid formulations
GB2551986A (en) 2016-07-01 2018-01-10 Gw Res Ltd Parenteral formulations
GB2559774B (en) 2017-02-17 2021-09-29 Gw Res Ltd Oral cannabinoid formulations
GB2569961B (en) 2018-01-03 2021-12-22 Gw Res Ltd Pharmaceutical

Citations (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0866073A1 (fr) * 1997-03-18 1998-09-23 Ajinomoto Co., Ltd. Nouveau dérivés dipeptidiques et agents édulcorantes
WO1999012957A1 (fr) * 1997-09-11 1999-03-18 The Nutrasweet Company SELS BASIQUES DE N-[N-(3,3-DIMETHYLBUTYL)-L-α-ASPARTYL]-L-PHENYLALANINE 1-METHYL ESTER
WO1999030576A1 (fr) * 1997-12-17 1999-06-24 The Nutrasweet Company Compositions de boissons comprenant un edulcorant presentant un tres fort pouvoir sucrant
JPH11279081A (ja) * 1998-03-27 1999-10-12 Ajinomoto Co Inc 苦味物質含有組成物
WO1999057998A1 (fr) * 1998-05-08 1999-11-18 Ajinomoto Co., Inc. Compositions a base d'edulcorants
WO1999062354A1 (fr) * 1998-06-05 1999-12-09 Wm. Wrigley Jr. Company Procede pour moduler la liberation de derives n-substitues d'aspartame dans une gomme a macher et gomme ainsi produite
WO2000036933A1 (fr) * 1998-12-18 2000-06-29 The Nutrasweet Company UTILISATION D'UN ESTER METHYLIQUE DE N-NEOHEXYL-$G(a)-ASPARTYL-L-PHENYLALANINE COMME AGENT DE SAPIDITE
WO2000057726A1 (fr) * 1999-03-29 2000-10-05 The Nutrasweet Company ALIMENTS FONCTIONNELS COMPRENANT UN ESTER DE 1-METHYLE N-[N-(3,3-DIMETHYLBUTYL)-L-α-ASPARTYL]-L-PHENYLALANINE

Patent Citations (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0866073A1 (fr) * 1997-03-18 1998-09-23 Ajinomoto Co., Ltd. Nouveau dérivés dipeptidiques et agents édulcorantes
WO1999012957A1 (fr) * 1997-09-11 1999-03-18 The Nutrasweet Company SELS BASIQUES DE N-[N-(3,3-DIMETHYLBUTYL)-L-α-ASPARTYL]-L-PHENYLALANINE 1-METHYL ESTER
WO1999030576A1 (fr) * 1997-12-17 1999-06-24 The Nutrasweet Company Compositions de boissons comprenant un edulcorant presentant un tres fort pouvoir sucrant
JPH11279081A (ja) * 1998-03-27 1999-10-12 Ajinomoto Co Inc 苦味物質含有組成物
WO1999057998A1 (fr) * 1998-05-08 1999-11-18 Ajinomoto Co., Inc. Compositions a base d'edulcorants
JPH11318381A (ja) * 1998-05-08 1999-11-24 Ajinomoto Co Inc 新規甘味料組成物
WO1999062354A1 (fr) * 1998-06-05 1999-12-09 Wm. Wrigley Jr. Company Procede pour moduler la liberation de derives n-substitues d'aspartame dans une gomme a macher et gomme ainsi produite
WO2000036933A1 (fr) * 1998-12-18 2000-06-29 The Nutrasweet Company UTILISATION D'UN ESTER METHYLIQUE DE N-NEOHEXYL-$G(a)-ASPARTYL-L-PHENYLALANINE COMME AGENT DE SAPIDITE
WO2000057726A1 (fr) * 1999-03-29 2000-10-05 The Nutrasweet Company ALIMENTS FONCTIONNELS COMPRENANT UN ESTER DE 1-METHYLE N-[N-(3,3-DIMETHYLBUTYL)-L-α-ASPARTYL]-L-PHENYLALANINE

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
DATABASE WPI Week 200006, Derwent World Patents Index; AN 2000-053011 *
PATENT ABSTRACTS OF JAPAN vol. 2000, no. 1 31 January 2000 (2000-01-31) *

Also Published As

Publication number Publication date
AU1093401A (en) 2001-04-30
WO2001028590A2 (fr) 2001-04-26

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