TN2010000351A1 - Novel hsp90 inhibitory carbazole derivatives compositions containing same and use thereof - Google Patents
Novel hsp90 inhibitory carbazole derivatives compositions containing same and use thereofInfo
- Publication number
- TN2010000351A1 TN2010000351A1 TNP2010000351A TN2010000351A TN2010000351A1 TN 2010000351 A1 TN2010000351 A1 TN 2010000351A1 TN P2010000351 A TNP2010000351 A TN P2010000351A TN 2010000351 A TN2010000351 A TN 2010000351A TN 2010000351 A1 TN2010000351 A1 TN 2010000351A1
- Authority
- TN
- Tunisia
- Prior art keywords
- alkyl
- compositions containing
- containing same
- carbazole derivatives
- optionally substituted
- Prior art date
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
The invention relates to the novel substances in Formula (I): wherein Het is a heterocycle optionally substituted by one or a plurality of radicals R1 or R'1; R is selected from the group comprising Formula (II) with R1 and/or R'1 selected from H, halogen, CF3, nitro, cyano, alkyl, hydroxyl, mercapto, amino, alkylamino, dialkylamino, alkoxy, phenylalcoxy, alkythio, or carboxy that is free or esterified by an alkyl, carboxamide, CO-NH(alkyl), CON(alkyl)2, NH-CO-alkyl, sulfonamide, NH-SO2-alkyl, S(O)2-NHalkyl, or S(O2)-N(alkyl)2 radical; all these radicals are optionally substituted; W1, W2, and W3 independently are CH or N; X is O, S, NR2, C(O), S(O), or S(O)2; Z is optionally substituted H, HaI, -O-R2 or –NH-R2 with R2 being H, alkyl, cycloalkyl, or heterocycloalkyl; and these substances are all isomeric forms and salts thereof, used as drugs.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/FR2009/000267 WO2009122034A2 (en) | 2008-03-14 | 2009-03-13 | Novel hsp90 inhibitory carbazole derivatives, compositions containing same, and use thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TN2010000351A1 true TN2010000351A1 (en) | 2011-12-29 |
Family
ID=55024481
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TNP2010000351A TN2010000351A1 (en) | 2009-03-13 | 2010-07-27 | Novel hsp90 inhibitory carbazole derivatives compositions containing same and use thereof |
Country Status (1)
| Country | Link |
|---|---|
| TN (1) | TN2010000351A1 (en) |
-
2010
- 2010-07-27 TN TNP2010000351A patent/TN2010000351A1/en unknown
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