IL165087A0 - New etonogestrel esters - Google Patents

New etonogestrel esters

Info

Publication number: IL165087A0
Authority: IL; Israel
Prior art keywords: new; etonogestrel esters; esters; new etonogestrel; etonogestrel
Prior art date: 2002-05-30

Application number

IL16508704A

Other languages

English (en)

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-05-30

Filing date

2004-11-08

Publication date

2005-12-18

2004-11-08 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

2005-12-18 Publication of IL165087A0 publication Critical patent/IL165087A0/xx

Links

GCKFUYQCUCGESZ-BPIQYHPVSA-N etonogestrel Chemical class O=C1CC[C@@H]2[C@H]3C(=C)C[C@](CC)([C@](CC4)(O)C#C)[C@@H]4[C@@H]3CCC2=C1 GCKFUYQCUCGESZ-BPIQYHPVSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- C07J1/0051—Estrane derivatives
- C07J1/0081—Substituted in position 17 alfa and 17 beta
- C07J1/0088—Substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
- C07J1/0096—Alkynyl derivatives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/16—Masculine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
- A61P5/34—Gestagens

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Endocrinology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Reproductive Health (AREA)
Diabetes (AREA)
Gynecology & Obstetrics (AREA)
Epidemiology (AREA)
Steroid Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

IL16508704A 2002-05-30 2004-11-08 New etonogestrel esters IL165087A0 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP02077119		2002-05-30
PCT/EP2003/050187 WO2003102012A2 (en)	2002-05-30	2003-05-22	New etonogestrel esters

Publications (1)

Publication Number	Publication Date
IL165087A0 true IL165087A0 (en)	2005-12-18

Family

ID=29595014

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
IL16508704A IL165087A0 (en)	2002-05-30	2004-11-08	New etonogestrel esters

Country Status (30)

Country	Link
US (1)	US7323454B2 (es)
EP (1)	EP1513861B1 (es)
JP (1)	JP4716726B2 (es)
KR (1)	KR20050009723A (es)
CN (2)	CN1314701C (es)
AR (1)	AR040130A1 (es)
AT (1)	ATE349458T1 (es)
AU (1)	AU2003238081B2 (es)
BR (1)	BR0311254A (es)
CA (1)	CA2487722C (es)
CO (1)	CO5631449A2 (es)
DE (1)	DE60310714T2 (es)
DK (1)	DK1513861T3 (es)
ES (1)	ES2277085T3 (es)
HR (1)	HRP20041101A2 (es)
IL (1)	IL165087A0 (es)
IS (1)	IS2421B (es)
MX (1)	MXPA04011797A (es)
NO (1)	NO20044898L (es)
NZ (1)	NZ536619A (es)
PE (1)	PE20040068A1 (es)
PL (1)	PL373855A1 (es)
PT (1)	PT1513861E (es)
RS (1)	RS97604A (es)
RU (1)	RU2325910C2 (es)
SI (1)	SI1513861T1 (es)
TW (1)	TW200403065A (es)
UA (1)	UA80126C2 (es)
WO (1)	WO2003102012A2 (es)
ZA (1)	ZA200410410B (es)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
TW200400041A (en) *	2002-05-30	2004-01-01	Akzo Nobel Nv	Use of new etonogestrel esters
US20090062909A1 (en)	2005-07-15	2009-03-05	Micell Technologies, Inc.	Stent with polymer coating containing amorphous rapamycin
WO2007011707A2 (en)	2005-07-15	2007-01-25	Micell Technologies, Inc.	Polymer coatings containing drug powder of controlled morphology
EP2944382A1 (en)	2006-04-26	2015-11-18	Micell Technologies, Inc.	Coatings containing multiple drugs
US11426494B2 (en)	2007-01-08	2022-08-30	MT Acquisition Holdings LLC	Stents having biodegradable layers
EP2111184B1 (en)	2007-01-08	2018-07-25	Micell Technologies, Inc.	Stents having biodegradable layers
US9433516B2 (en)	2007-04-17	2016-09-06	Micell Technologies, Inc.	Stents having controlled elution
MX350637B (es)	2008-04-17	2017-09-11	Micell Technologies Inc	Stents que tienen capas bioabsorbibles.
JP2011528275A (ja)	2008-07-17	2011-11-17	ミセルテクノロジーズ，インク．	薬物送達医療デバイス
WO2010111232A2 (en)	2009-03-23	2010-09-30	Micell Technologies, Inc.	Drug delivery medical device
US9981072B2 (en)	2009-04-01	2018-05-29	Micell Technologies, Inc.	Coated stents
EP2453834A4 (en)	2009-07-16	2014-04-16	Micell Technologies Inc	MEDICAL DEVICE DISPENSING MEDICINE
EP2531140B1 (en)	2010-02-02	2017-11-01	Micell Technologies, Inc.	Stent and stent delivery system with improved deliverability
WO2011133655A1 (en)	2010-04-22	2011-10-27	Micell Technologies, Inc.	Stents and other devices having extracellular matrix coating
EP2593039B1 (en)	2010-07-16	2022-11-30	Micell Technologies, Inc.	Drug delivery medical device
US10117972B2 (en)	2011-07-15	2018-11-06	Micell Technologies, Inc.	Drug delivery medical device
US10188772B2 (en)	2011-10-18	2019-01-29	Micell Technologies, Inc.	Drug delivery medical device
JP6330024B2 (ja)	2013-03-12	2018-05-23	マイセル・テクノロジーズ，インコーポレイテッド	生体吸収性バイオメディカルインプラント
KR20180059584A (ko)	2013-05-15	2018-06-04	미셀 테크놀로지즈, 인코포레이티드	생흡수성 생체의학적 임플란트
RU2595818C1 (ru) *	2015-05-25	2016-08-27	Федеральное государственное бюджетное научное учреждение "Научный центр проблем здоровья семьи и репродукции человека"	Способ комплексного лечения дисфункции яичников при применении гормонального контрацептива имплантата "импланона"
CN111057120B (zh) *	2019-12-27	2021-04-27	苏州翔实医药发展有限公司	一种依托孕烯衍生物a及其制备方法和用途

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB845442A (en)	1956-03-22	1960-08-24	Schering Ag	Manufacture of steroid compounds
DE1013284B (de)	1956-03-22	1957-08-08	Schering Ag	Verfahren zur Einfuehrung der Reste wenig reaktionsfaehiger Carbonsaeuren, insbesondere des ª‰-Cyclopentyl-propionylrestes, in die 17ª‡-staendige Oxygruppe solcher Steroide, die am Kohlenstoffatom 17 neben der Oxygruppe eine Acetylgruppe tragen
GB8313921D0 (en) *	1983-05-19	1983-06-22	World Health Org	Contraceptive compositions
DE4227989A1 (de)	1992-08-21	1994-06-09	Schering Ag	Mittel zur transdermalen Applikation enthaltend 3-Keto-desogestrel
DE4240806A1 (de)	1992-12-01	1994-06-09	Schering Ag	Mittel zur transdermalen Applikation enthaltend 14alpha,17alpha-Ethanoestra-1,3,5(10)-trien-3,17beta-diol
JPH07101884A (ja)	1993-10-01	1995-04-18	Sanei Gen F F I Inc	水溶性ヘミセルロースを含有する製剤
NZ277552A (en) *	1993-12-27	1998-01-26	Akzo Nobel Nv	Steroid preparation which is percutaneously absorbable
DE19613698A1 (de)	1995-07-17	1997-01-23	Schering Ag	Mittel zur transdermalen Applikation enthaltend Ester des 13-Ethyl-17ß-hydroxy-11-methylen-18,19-dinor-17alpha-pregn-4-en-20-yn-3-ons
JPH11509222A (ja) *	1995-07-17	1999-08-17	シェリングアクチェンゲゼルシャフト	１３−エチル−１７β−ヒドロキシ−１１−メチレン−１８，１９−ジノル−１７α−プレグン−４−エン−２０−イン−３−オンのエステルを含む経皮投与のための剤
DE19531936A1 (de) *	1995-08-17	1997-02-20	Schering Ag	Kombinationspräparat zur Kontrazeption, Kits diese enthaltend und eine Methode diese verwendend
DE19540253C2 (de) *	1995-10-28	1998-06-04	Jenapharm Gmbh	Mehrphasenpräparat zur Kontrazeption auf der Basis natürlicher Estrogene
DK1087986T3 (da)	1998-06-19	2002-06-17	Akzo Nobel Nv	Testosteronderivat
AU4513099A (en)	1998-06-19	2000-01-10	Akzo Nobel N.V.	Cycloalkyl-carboxylic acid esters of 7.alpha.methyl-estr-4-en-3-one 17.beta.-ol (19-nor 7.alpha.-methyltestosterone)
US6180682B1 (en)	1999-01-26	2001-01-30	Virgil A. Place	Buccal drug delivery system for use in male contraception
TW200400041A (en) *	2002-05-30	2004-01-01	Akzo Nobel Nv	Use of new etonogestrel esters

2003
- 2003-05-19 TW TW092113489A patent/TW200403065A/zh unknown
- 2003-05-22 PT PT03735713T patent/PT1513861E/pt unknown
- 2003-05-22 MX MXPA04011797A patent/MXPA04011797A/es active IP Right Grant
- 2003-05-22 KR KR10-2004-7019330A patent/KR20050009723A/ko not_active Ceased
- 2003-05-22 CA CA2487722A patent/CA2487722C/en not_active Expired - Fee Related
- 2003-05-22 PL PL03373855A patent/PL373855A1/xx unknown
- 2003-05-22 CN CNB038123754A patent/CN1314701C/zh not_active Expired - Fee Related
- 2003-05-22 ES ES03735713T patent/ES2277085T3/es not_active Expired - Lifetime
- 2003-05-22 RS YU97604A patent/RS97604A/sr unknown
- 2003-05-22 NZ NZ536619A patent/NZ536619A/en unknown
- 2003-05-22 HR HRP20041101 patent/HRP20041101A2/xx not_active Application Discontinuation
- 2003-05-22 DE DE60310714T patent/DE60310714T2/de not_active Expired - Lifetime
- 2003-05-22 DK DK03735713T patent/DK1513861T3/da active
- 2003-05-22 US US10/516,402 patent/US7323454B2/en not_active Expired - Lifetime
- 2003-05-22 WO PCT/EP2003/050187 patent/WO2003102012A2/en active IP Right Grant
- 2003-05-22 RU RU2004138807/15A patent/RU2325910C2/ru not_active IP Right Cessation
- 2003-05-22 CN CNA2007101028610A patent/CN101100480A/zh active Pending
- 2003-05-22 AT AT03735713T patent/ATE349458T1/de not_active IP Right Cessation
- 2003-05-22 SI SI200330679T patent/SI1513861T1/sl unknown
- 2003-05-22 UA UA20041109287A patent/UA80126C2/uk unknown
- 2003-05-22 BR BR0311254-3A patent/BR0311254A/pt not_active IP Right Cessation
- 2003-05-22 EP EP03735713A patent/EP1513861B1/en not_active Expired - Lifetime
- 2003-05-22 JP JP2004509703A patent/JP4716726B2/ja not_active Expired - Fee Related
- 2003-05-22 AU AU2003238081A patent/AU2003238081B2/en not_active Ceased
- 2003-05-28 PE PE2003000517A patent/PE20040068A1/es not_active Application Discontinuation
- 2003-05-28 AR ARP030101859A patent/AR040130A1/es unknown
2004
- 2004-11-08 IL IL16508704A patent/IL165087A0/xx unknown
- 2004-11-10 NO NO20044898A patent/NO20044898L/no not_active Application Discontinuation
- 2004-11-15 IS IS7528A patent/IS2421B/is unknown
- 2004-12-22 CO CO04127949A patent/CO5631449A2/es not_active Application Discontinuation
- 2004-12-23 ZA ZA200410410A patent/ZA200410410B/xx unknown

Also Published As

Publication number	Publication date
JP2005532350A (ja)	2005-10-27
TW200403065A (en)	2004-03-01
CN1692122A (zh)	2005-11-02
WO2003102012A2 (en)	2003-12-11
BR0311254A (pt)	2005-03-15
WO2003102012A3 (en)	2004-04-22
MXPA04011797A (es)	2005-03-31
CA2487722C (en)	2011-07-19
DE60310714T2 (de)	2007-10-11
KR20050009723A (ko)	2005-01-25
US20050222113A1 (en)	2005-10-06
DK1513861T3 (da)	2007-04-10
ES2277085T3 (es)	2007-07-01
AU2003238081B2 (en)	2008-09-18
CA2487722A1 (en)	2003-12-11
HK1072609A1 (en)	2005-09-02
PT1513861E (pt)	2007-03-30
CN101100480A (zh)	2008-01-09
ZA200410410B (en)	2006-02-22
PL373855A1 (en)	2005-09-19
US7323454B2 (en)	2008-01-29
SI1513861T1 (sl)	2007-06-30
RU2004138807A (ru)	2005-05-27
UA80126C2 (en)	2007-08-27
EP1513861A2 (en)	2005-03-16
WO2003102012A9 (en)	2005-01-13
AR040130A1 (es)	2005-03-16
ATE349458T1 (de)	2007-01-15
PE20040068A1 (es)	2004-02-18
EP1513861B1 (en)	2006-12-27
IS7528A (is)	2004-11-15
AU2003238081A1 (en)	2003-12-19
IS2421B (is)	2008-10-15
NO20044898L (no)	2005-02-25
CN1314701C (zh)	2007-05-09
RS97604A (en)	2006-10-27
JP4716726B2 (ja)	2011-07-06
DE60310714D1 (de)	2007-02-08
RU2325910C2 (ru)	2008-06-10
CO5631449A2 (es)	2006-04-28
HRP20041101A2 (en)	2004-12-31
NZ536619A (en)	2007-09-28

Publication	Publication Date	Title
AU2003249738A8 (en)	2004-01-23	Ostoscope
AU2003297193A8 (en)	2004-07-09	Meta-web
IL165087A0 (en)	2005-12-18	New etonogestrel esters
AU2003252028A8 (en)	2004-02-09	Heterodiamondoids
AU2003279495A8 (en)	2004-05-13	Alert-modeling
GB2400797B (en)	2006-12-20	Shelving
AU2003264900A8 (en)	2004-04-08	Cast-cutter
AU2002367810A8 (en)	2003-11-10	Bis-transition-metal-chelate-probes
IL165125A0 (en)	2005-12-18	Use of new etonogestrel esters
AU2003262681A8 (en)	2004-03-03	Hemo-aide
GB0310123D0 (en)	2003-06-04	Airfreshener combined luminair
AU2002341221A8 (en)	2004-04-19	Honey-brandy
AU2003253735A8 (en)	2004-01-06	Vacuolins
GB0215011D0 (en)	2002-08-07	Easy squeezy
GB0204882D0 (en)	2002-04-17	Pedestal
AU2328P (en)	2003-09-25	Archley Arctotis fastuosa
AU2327P (en)	2003-09-25	Archnah Arctotis fastuosa
AU2326P (en)	2003-09-25	Gavol Gazania rigens
AU150609S (en)	2003-02-11	Weephole former
PL113111U1 (en)	2003-10-06	Shelving
GB0214885D0 (en)	2002-08-07	Medicament
GB0211377D0 (en)	2002-06-26	Medicament
GB0227620D0 (en)	2003-01-08	Easy Klik
GB0210565D0 (en)	2002-06-19	Concept three
AU149787S (en)	2002-11-06	Pedestal