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DK0526543T3 - Derivater og analoger af 2-deoxy-2,3-didehydro-N-acetylneuraminsyre og deres anvendelse som antivirale midler - Google Patents

Derivater og analoger af 2-deoxy-2,3-didehydro-N-acetylneuraminsyre og deres anvendelse som antivirale midler

Info

Publication number
DK0526543T3
DK0526543T3 DK91908682T DK91908682T DK0526543T3 DK 0526543 T3 DK0526543 T3 DK 0526543T3 DK 91908682 T DK91908682 T DK 91908682T DK 91908682 T DK91908682 T DK 91908682T DK 0526543 T3 DK0526543 T3 DK 0526543T3
Authority
DK
Denmark
Prior art keywords
didehydro
antivirals
deoxy
analogues
derivatives
Prior art date
Application number
DK91908682T
Other languages
Danish (da)
English (en)
Inventor
Itzstein Laurence Mark Von
Wen-Yang Wu
Tho Van Phan
Basil Danylec
Betty Jin
Peter Malcolm Colman
Joseph Noozhumurry Varghese
Original Assignee
Biota Scient Management
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Biota Scient Management filed Critical Biota Scient Management
Application granted granted Critical
Publication of DK0526543T3 publication Critical patent/DK0526543T3/da

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D309/30Oxygen atoms, e.g. delta-lactones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Virology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Compounds Containing Sulfur Atoms (AREA)
  • Hydrogenated Pyridines (AREA)
  • Pyrane Compounds (AREA)
DK91908682T 1990-04-24 1991-04-24 Derivater og analoger af 2-deoxy-2,3-didehydro-N-acetylneuraminsyre og deres anvendelse som antivirale midler DK0526543T3 (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
AUPJ980090 1990-04-24
AUPK289690 1990-10-19
AUPK453791 1991-02-11
PCT/AU1991/000161 WO1991016320A1 (fr) 1990-04-24 1991-04-24 Derives et analogues d'acide 2-deoxy-2,3-didehydro-n-acetyle neuraminique et leur utilisation comme agents antiviraux

Publications (1)

Publication Number Publication Date
DK0526543T3 true DK0526543T3 (da) 1998-08-24

Family

ID=27157556

Family Applications (1)

Application Number Title Priority Date Filing Date
DK91908682T DK0526543T3 (da) 1990-04-24 1991-04-24 Derivater og analoger af 2-deoxy-2,3-didehydro-N-acetylneuraminsyre og deres anvendelse som antivirale midler

Country Status (37)

Country Link
US (2) US5360817A (fr)
EP (2) EP0786458B1 (fr)
JP (1) JP2944750B2 (fr)
KR (1) KR0169496B1 (fr)
CN (3) CN1036849C (fr)
AP (1) AP249A (fr)
AT (2) ATE161253T1 (fr)
AU (2) AU654815B2 (fr)
BG (1) BG62092B1 (fr)
CA (2) CA2081356C (fr)
CY (1) CY2186B1 (fr)
CZ (1) CZ288492B6 (fr)
DE (3) DE19975068I2 (fr)
DK (1) DK0526543T3 (fr)
ES (2) ES2113881T3 (fr)
FI (2) FI105478B (fr)
GR (1) GR3026225T3 (fr)
HK (2) HK1003834A1 (fr)
HU (2) HU219355B (fr)
IE (2) IE911372A1 (fr)
IL (1) IL97936A (fr)
LU (1) LU90468I2 (fr)
MY (1) MY107843A (fr)
NL (1) NL990030I2 (fr)
NO (3) NO302751B1 (fr)
NZ (1) NZ237936A (fr)
OA (1) OA09679A (fr)
PL (3) PL167630B1 (fr)
PT (1) PT97460B (fr)
RU (1) RU2119487C1 (fr)
SG (1) SG43170A1 (fr)
SI (1) SI9110745B (fr)
SK (1) SK282950B6 (fr)
UA (1) UA41252C2 (fr)
WO (1) WO1991016320A1 (fr)
YU (1) YU48741B (fr)
ZA (1) ZA913086B (fr)

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* Cited by examiner, † Cited by third party
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TWI764917B (zh) 2016-08-22 2022-05-21 醣基生醫股份有限公司 抗體、結合片段及使用方法
CN106520864A (zh) * 2016-09-28 2017-03-22 南京农业大学 一种酶法合成唾液酸类似物的方法及其应用
AU2018273411B2 (en) * 2017-05-25 2022-12-01 The Governors Of The University Of Alberta Methods of preventing or treating atherosclerosis with inhibitors of specific isoenzymes of human neuraminidase
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