CL2007003765A1 - COMPOUNDS DERIVED FROM 2-OXO-4-HIDROXI-BENZOTIAZOL; PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION; PHARMACEUTICAL COMBINATION; AND USE IN THE TREATMENT OF DISEASES SUCH AS COPD, BRONCHITIS, ASTHMA AND BRONCHIECTASIES. - Google Patents
COMPOUNDS DERIVED FROM 2-OXO-4-HIDROXI-BENZOTIAZOL; PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION; PHARMACEUTICAL COMBINATION; AND USE IN THE TREATMENT OF DISEASES SUCH AS COPD, BRONCHITIS, ASTHMA AND BRONCHIECTASIES.Info
- Publication number
- CL2007003765A1 CL2007003765A1 CL200703765A CL2007003765A CL2007003765A1 CL 2007003765 A1 CL2007003765 A1 CL 2007003765A1 CL 200703765 A CL200703765 A CL 200703765A CL 2007003765 A CL2007003765 A CL 2007003765A CL 2007003765 A1 CL2007003765 A1 CL 2007003765A1
- Authority
- CL
- Chile
- Prior art keywords
- bronchiectasies
- benzotiazol
- hidroxi
- copd
- bronchitis
- Prior art date
Links
- 208000006545 Chronic Obstructive Pulmonary Disease Diseases 0.000 title 1
- 208000006673 asthma Diseases 0.000 title 1
- 206010006451 bronchitis Diseases 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 201000010099 disease Diseases 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 238000002360 preparation method Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/08—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D277/12—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/14—Oxygen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/14—Thiadiazoles; Hydrogenated thiadiazoles condensed with carbocyclic rings or ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Otolaryngology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Plural Heterocyclic Compounds (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US87092206P | 2006-12-20 | 2006-12-20 | |
US91004507P | 2007-04-04 | 2007-04-04 | |
US95198007P | 2007-07-26 | 2007-07-26 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2007003765A1 true CL2007003765A1 (en) | 2008-08-22 |
Family
ID=39167020
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL200703765A CL2007003765A1 (en) | 2006-12-20 | 2007-12-20 | COMPOUNDS DERIVED FROM 2-OXO-4-HIDROXI-BENZOTIAZOL; PREPARATION PROCESS; PHARMACEUTICAL COMPOSITION; PHARMACEUTICAL COMBINATION; AND USE IN THE TREATMENT OF DISEASES SUCH AS COPD, BRONCHITIS, ASTHMA AND BRONCHIECTASIES. |
Country Status (21)
Country | Link |
---|---|
US (3) | US7700782B2 (en) |
EP (1) | EP2121642B1 (en) |
JP (1) | JP2010513440A (en) |
KR (1) | KR20090091342A (en) |
AR (1) | AR064635A1 (en) |
AT (1) | ATE517879T1 (en) |
AU (1) | AU2007336075B2 (en) |
BR (1) | BRPI0722096A2 (en) |
CA (1) | CA2672811A1 (en) |
CL (1) | CL2007003765A1 (en) |
CO (1) | CO6190554A2 (en) |
EC (1) | ECSP099426A (en) |
HK (1) | HK1136572A1 (en) |
IL (1) | IL199014A0 (en) |
MX (1) | MX2009006009A (en) |
NO (1) | NO20092691L (en) |
PE (1) | PE20081544A1 (en) |
SA (1) | SA07280728B1 (en) |
TW (1) | TW200833670A (en) |
UY (1) | UY30808A1 (en) |
WO (1) | WO2008075026A1 (en) |
Families Citing this family (17)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
TW200738658A (en) * | 2005-08-09 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
TW200738659A (en) * | 2005-08-29 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
TW200745067A (en) * | 2006-03-14 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
TW200825084A (en) | 2006-11-14 | 2008-06-16 | Astrazeneca Ab | New compounds 521 |
TW200833670A (en) * | 2006-12-20 | 2008-08-16 | Astrazeneca Ab | Novel compounds 569 |
GB0702458D0 (en) * | 2007-02-08 | 2007-03-21 | Astrazeneca Ab | Salts 668 |
CN102088976B (en) * | 2008-05-13 | 2012-12-26 | 阿斯利康(瑞典)有限公司 | Pharmaceutical product comprising a muscarinic receptor antagonist and a beta2-adrenoceptor agonist |
EA017627B1 (en) | 2008-05-13 | 2013-01-30 | Астразенека Аб | Quinuclidine derivatives as muscarinic m3 receptor antagonists |
AU2009260899B2 (en) | 2008-06-18 | 2012-02-23 | Astrazeneca Ab | Benzoxazinone derivatives acting as beta2-adrenoreceptor agonist for the treatment of respiratory disorders |
KR20110022611A (en) * | 2008-06-20 | 2011-03-07 | 아스트라제네카 아베 | Pharmaceutical composition comprising 4-hydroxy-2-oxo-2,3-dihydro-1,3-benzothiazol-7-yl compound for the regulation of beta-2-adrenergic receptor activity |
GB0814728D0 (en) * | 2008-08-12 | 2008-09-17 | Argenta Discovery Ltd | New combination |
TW201036957A (en) | 2009-02-20 | 2010-10-16 | Astrazeneca Ab | Novel salt 628 |
GB0913342D0 (en) | 2009-07-31 | 2009-09-16 | Astrazeneca Ab | Compounds - 801 |
WO2011061527A1 (en) | 2009-11-17 | 2011-05-26 | Astrazeneca Ab | Combinations comprising a glucocorticoid receptor modulator for the treatment of respiratory diseases |
GB201016912D0 (en) | 2010-10-07 | 2010-11-24 | Astrazeneca Ab | Novel combination |
JO3192B1 (en) | 2011-09-06 | 2018-03-08 | Novartis Ag | Benzothiazolone compound |
WO2015050984A1 (en) * | 2013-10-01 | 2015-04-09 | New York University | Amino, amido, and heterocyclic compounds as modulators of rage activity and uses thereof |
Family Cites Families (76)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2653977A (en) * | 1953-09-29 | Chxnx | ||
US3775477A (en) * | 1971-03-10 | 1973-11-27 | Sterling Drug Inc | N,n'-bis(2-aryl-2-(hydroxy or oxo)-ethyl)-bridged-bis-carboxamides |
US4460581A (en) * | 1982-10-12 | 1984-07-17 | Boehringer Ingelheim Kg | (1-Hydroxy-2-amino-alkyl)-substituted benzoxazinones and benzoxazolinones |
DE3571808D1 (en) | 1984-04-17 | 1989-08-31 | Glaxo Group Ltd | Ethanolamine compounds |
US4554284A (en) | 1984-09-12 | 1985-11-19 | Smithkline Beckman Corporation | 7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones |
US4554287A (en) | 1984-09-12 | 1985-11-19 | Smithkline Beckman Corporation | Antihypertensive 7-[2-(dialkylamino)ethyl]-4-hydroxy-1,3-benzimidazol-2-ones |
GB8525483D0 (en) | 1985-10-16 | 1985-11-20 | Glaxo Group Ltd | Chemical compounds |
GB8718938D0 (en) | 1987-08-11 | 1987-09-16 | Glaxo Group Ltd | Chemical compounds |
EP0422889A3 (en) | 1989-10-10 | 1991-08-28 | Glaxo Group Limited | Phenethanolamine compounds |
GB9210632D0 (en) | 1992-05-19 | 1992-07-01 | Fisons Plc | Compounds |
US5648370A (en) * | 1990-11-20 | 1997-07-15 | Astra Pharmaceuticals Limited | 7-(2-aminoethyl) benzothiazolones |
GB9211172D0 (en) | 1992-05-27 | 1992-07-08 | Fisons Plc | Compounds |
IE914003A1 (en) | 1990-11-20 | 1992-05-20 | Astra Pharma Prod | Biologically Active Amines |
TW356468B (en) * | 1995-09-15 | 1999-04-21 | Astra Pharma Prod | Benzothiazolone compounds useful as beta2-adrenoreceptor and dopamine DA2 receptor agonists process for preparing same and pharmaceutical compositions containing same |
GB9526511D0 (en) | 1995-12-23 | 1996-02-28 | Astra Pharma Prod | Pharmaceutically active compounds |
DE69709647T2 (en) | 1996-05-20 | 2002-11-07 | Dupont Pharmaceuticals Research Laboratories, Inc. | CYCLIC DIARYLALKYL DIAMINE DERIVATIVES AS AN ANTOGONISTS OF CHEMOKINE RECEPTORS |
SE9700706D0 (en) | 1997-02-27 | 1997-02-27 | Astra Pharma Prod | Process for the preparation of benzothiazoline compounds |
SE9701304D0 (en) | 1997-04-09 | 1997-04-09 | Astra Pharma Prod | Compounds |
EP1075278A1 (en) | 1998-01-13 | 2001-02-14 | AstraZeneca UK Limited | PHARMACEUTICAL COMPOSITIONS COMPRISING A COMPOUND HAVING DOPAMINE (D 2?) RECEPTOR AGONIST ACTIVITY AND A COMPOUND (B) HAVING $g(b) 2?-ADRENORECEPTOR AGONIST ACTIVITY |
US6541669B1 (en) | 1998-06-08 | 2003-04-01 | Theravance, Inc. | β2-adrenergic receptor agonists |
GB9913083D0 (en) | 1999-06-04 | 1999-08-04 | Novartis Ag | Organic compounds |
US6683115B2 (en) * | 1999-06-02 | 2004-01-27 | Theravance, Inc. | β2-adrenergic receptor agonists |
SE9902937D0 (en) | 1999-08-18 | 1999-08-18 | Astra Pharma Prod | Pharmaceutical compositions |
SE9902936D0 (en) | 1999-08-18 | 1999-08-18 | Astra Pharma Prod | Pharmaceutical compositions |
SE9902938D0 (en) | 1999-08-18 | 1999-08-18 | Astra Pharma Prod | Pharmaceutical compositions |
SE9902935D0 (en) | 1999-08-18 | 1999-08-18 | Astra Pharma Prod | Pharmaceutical compositions |
OA11558A (en) | 1999-12-08 | 2004-06-03 | Advanced Medicine Inc | Beta 2-adrenergic receptor agonists. |
US6506901B2 (en) | 2000-07-17 | 2003-01-14 | Wyeth | Substituted 2-(S)-hydroxy-3-(piperidin-4-yl-methylamino)-propyl ethers and substituted 2-aryl-2-(R)-hydroxy-1-(piperidin-4-yl-methyl)-ethylamine β-3 adrenergic receptor agonists |
US7045658B2 (en) | 2001-03-22 | 2006-05-16 | Glaxo Group Limited | Formailide derivatives as beta2-adrenoreceptor agonists |
KR100912324B1 (en) | 2001-09-14 | 2009-08-14 | 글락소 그룹 리미티드 | Penethanolamine Derivatives for the Treatment of Respiratory Diseases |
US20030229058A1 (en) * | 2001-11-13 | 2003-12-11 | Moran Edmund J. | Aryl aniline beta2 adrenergic receptor agonists |
GB0217225D0 (en) | 2002-07-25 | 2002-09-04 | Glaxo Group Ltd | Medicinal compounds |
AR040962A1 (en) * | 2002-08-09 | 2005-04-27 | Novartis Ag | COMPOUNDS DERIVED FROM TIAZOL 1,3-2-ONA, PHARMACEUTICAL COMPOSITION AND COMPOSITE PREPARATION PROCESS |
GB0225540D0 (en) | 2002-11-01 | 2002-12-11 | Glaxo Group Ltd | Medicinal compounds |
PE20040950A1 (en) | 2003-02-14 | 2005-01-01 | Theravance Inc | BIPHENYL DERIVATIVES AS AGONISTS OF ß2-ADRENERGIC RECEPTORS AND AS ANTAGONISTS OF MUSCARINAL RECEPTORS |
GB0303396D0 (en) | 2003-02-14 | 2003-03-19 | Glaxo Group Ltd | Medicinal compounds |
EP1615881A2 (en) | 2003-04-01 | 2006-01-18 | Theravance, Inc. | Diarylmethyl and related compounds having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity |
TW200526547A (en) | 2003-09-22 | 2005-08-16 | Theravance Inc | Amino-substituted ethylamino β2 adrenergic receptor agonists |
GB0324654D0 (en) | 2003-10-22 | 2003-11-26 | Glaxo Group Ltd | Medicinal compounds |
GB0324886D0 (en) | 2003-10-24 | 2003-11-26 | Glaxo Group Ltd | Medicinal compounds |
JP2005187357A (en) | 2003-12-25 | 2005-07-14 | Nippon Suisan Kaisha Ltd | METHOD FOR PRODUCING BENZOTHIAZOLONE DERIVATIVE HAVING SELECTIVE beta2-RECEPTOR AGONIST ACTIVITY |
TW200531692A (en) | 2004-01-12 | 2005-10-01 | Theravance Inc | Aryl aniline derivatives as β2 adrenergic receptor agonists |
GB0402797D0 (en) | 2004-02-09 | 2004-03-10 | Novartis Ag | Organic compounds |
WO2005092861A1 (en) | 2004-03-11 | 2005-10-06 | Pfizer Limited | Quinolinone derivatives pharmaceutical compositions containing them and their use |
EP1577306A1 (en) | 2004-03-17 | 2005-09-21 | Boehringer Ingelheim Pharma GmbH & Co.KG | novel benzoxazinone derivatives as slow-acting betamimetics and use thereof in treatment of respiratory tract diseases |
WO2005092841A1 (en) | 2004-03-23 | 2005-10-06 | Pfizer Limited | Compounds having beta-agonist activity |
JP2007537187A (en) | 2004-05-13 | 2007-12-20 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | Hydroxy-substituted benzofused heterocyclic compounds for use as beta agonists in the treatment of respiratory diseases |
EP1595873A1 (en) | 2004-05-13 | 2005-11-16 | Boehringer Ingelheim Pharma GmbH & Co.KG | Substituted cycloalkyl derivatives for the treatment of respiratory diseases |
DE102004024453A1 (en) | 2004-05-14 | 2006-01-05 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | New long-acting bronchodilators for the treatment of respiratory diseases |
US20080039495A1 (en) | 2004-06-03 | 2008-02-14 | Linsell Martin S | Diamine Beta2 Adrenergic Receptor Agonists |
EP1778638A1 (en) | 2004-07-21 | 2007-05-02 | Theravance, Inc. | Diaryl ether beta2 adrenergic receptor agonists |
EP1778626A1 (en) | 2004-08-16 | 2007-05-02 | Theravance, Inc. | Compounds having beta2 adrenergic receptor agonist and muscarinic receptor antagonist activity |
WO2006023460A2 (en) | 2004-08-16 | 2006-03-02 | Theravance, Inc. | COMPOUNDS HAVING β2 ADRENERGIC RECEPTOR AGONIST AND MUSCARINIC RECEPTOR ANTAGONIST ACTIVITY |
US7566785B2 (en) | 2004-09-10 | 2009-07-28 | Theravance, Inc. | Amidine substituted aryl aniline compounds |
GB0426164D0 (en) | 2004-11-29 | 2004-12-29 | Novartis Ag | Organic compounds |
WO2006074897A1 (en) | 2005-01-11 | 2006-07-20 | Glaxo Group Limited | Cinnamate salts of a beta-2 adrenergic agonist |
GB0511066D0 (en) | 2005-05-31 | 2005-07-06 | Novartis Ag | Organic compounds |
CA2614757C (en) | 2005-07-18 | 2011-11-08 | Pfizer Limited | Process for the preparation of sulfonamide derivatives |
TW200738658A (en) * | 2005-08-09 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
TW200740781A (en) | 2005-08-29 | 2007-11-01 | Astrazeneca Ab | Novel compounds |
TW200738659A (en) * | 2005-08-29 | 2007-10-16 | Astrazeneca Ab | Novel compounds |
US20090029958A1 (en) * | 2006-03-08 | 2009-01-29 | Lilian Alcaraz | Phenethanolamine derivatives as beta2 adrenoreceptor agonists |
TW200745084A (en) | 2006-03-08 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
TW200745067A (en) | 2006-03-14 | 2007-12-16 | Astrazeneca Ab | Novel compounds |
WO2008041914A1 (en) | 2006-10-06 | 2008-04-10 | Astrazeneca Ab | 5-(2-AMINO-L-HYDROXYETHYL)-8-HYDROXY-2-OXOQUINOLINE DERIVATIVES AND OTHER COMPOUNDS AS β2 -ADRENERGIC AGONISTS |
TW200833670A (en) | 2006-12-20 | 2008-08-16 | Astrazeneca Ab | Novel compounds 569 |
US20120142646A1 (en) | 2006-12-20 | 2012-06-07 | Lilian Alcaraz | Novel Compounds 621 |
GB0702456D0 (en) | 2007-02-08 | 2007-03-21 | Astrazeneca Ab | New combination |
GB0702458D0 (en) * | 2007-02-08 | 2007-03-21 | Astrazeneca Ab | Salts 668 |
GB0702457D0 (en) | 2007-02-08 | 2007-03-21 | Astrazeneca Ab | New combination 666 |
GB0702459D0 (en) | 2007-02-08 | 2007-03-21 | Astrazeneca Ab | Salts 669 |
GB0703999D0 (en) | 2007-03-01 | 2007-04-11 | Astrazeneca Ab | New combination 667 |
GB0704000D0 (en) | 2007-03-01 | 2007-04-11 | Astrazeneca Ab | Salts 670 |
WO2009037503A2 (en) | 2007-09-18 | 2009-03-26 | Astrazeneca Ab | New combination - 012 for the treatment of respiratory diseases |
JP5646341B2 (en) * | 2007-12-20 | 2014-12-24 | アストラゼネカ・アクチエボラーグAstrazeneca Aktiebolag | Dosage device and method for mixing powder in airflow 537 |
KR20110022611A (en) * | 2008-06-20 | 2011-03-07 | 아스트라제네카 아베 | Pharmaceutical composition comprising 4-hydroxy-2-oxo-2,3-dihydro-1,3-benzothiazol-7-yl compound for the regulation of beta-2-adrenergic receptor activity |
-
2007
- 2007-12-07 TW TW096146813A patent/TW200833670A/en unknown
- 2007-12-19 WO PCT/GB2007/004861 patent/WO2008075026A1/en active Application Filing
- 2007-12-19 US US11/959,679 patent/US7700782B2/en not_active Expired - Fee Related
- 2007-12-19 JP JP2009542202A patent/JP2010513440A/en active Pending
- 2007-12-19 UY UY30808A patent/UY30808A1/en unknown
- 2007-12-19 BR BRPI0722096-0A2A patent/BRPI0722096A2/en not_active IP Right Cessation
- 2007-12-19 AU AU2007336075A patent/AU2007336075B2/en not_active Ceased
- 2007-12-19 AT AT07848598T patent/ATE517879T1/en not_active IP Right Cessation
- 2007-12-19 US US12/519,552 patent/US20100022491A1/en not_active Abandoned
- 2007-12-19 MX MX2009006009A patent/MX2009006009A/en active IP Right Grant
- 2007-12-19 CA CA002672811A patent/CA2672811A1/en not_active Abandoned
- 2007-12-19 KR KR1020097015062A patent/KR20090091342A/en not_active Withdrawn
- 2007-12-19 EP EP07848598A patent/EP2121642B1/en active Active
- 2007-12-20 AR ARP070105801A patent/AR064635A1/en not_active Application Discontinuation
- 2007-12-20 CL CL200703765A patent/CL2007003765A1/en unknown
- 2007-12-29 SA SA7280728A patent/SA07280728B1/en unknown
-
2008
- 2008-01-02 PE PE2008000009A patent/PE20081544A1/en not_active Application Discontinuation
-
2009
- 2009-05-27 CO CO09054440A patent/CO6190554A2/en not_active Application Discontinuation
- 2009-05-27 IL IL199014A patent/IL199014A0/en unknown
- 2009-06-15 EC EC2009009426A patent/ECSP099426A/en unknown
- 2009-07-15 NO NO20092691A patent/NO20092691L/en not_active Application Discontinuation
-
2010
- 2010-03-30 US US12/750,014 patent/US20100249200A1/en not_active Abandoned
- 2010-04-24 HK HK10104038.4A patent/HK1136572A1/en not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
EP2121642A1 (en) | 2009-11-25 |
PE20081544A1 (en) | 2009-01-11 |
CA2672811A1 (en) | 2008-06-26 |
US20100249200A1 (en) | 2010-09-30 |
BRPI0722096A2 (en) | 2014-04-01 |
NO20092691L (en) | 2009-09-16 |
US20100022491A1 (en) | 2010-01-28 |
US7700782B2 (en) | 2010-04-20 |
SA07280728B1 (en) | 2010-12-01 |
US20080207698A1 (en) | 2008-08-28 |
IL199014A0 (en) | 2010-02-17 |
AU2007336075A1 (en) | 2008-06-26 |
WO2008075026A1 (en) | 2008-06-26 |
ECSP099426A (en) | 2009-07-31 |
ATE517879T1 (en) | 2011-08-15 |
TW200833670A (en) | 2008-08-16 |
HK1136572A1 (en) | 2010-07-02 |
AU2007336075B2 (en) | 2011-10-27 |
MX2009006009A (en) | 2009-06-16 |
KR20090091342A (en) | 2009-08-27 |
CO6190554A2 (en) | 2010-08-19 |
AR064635A1 (en) | 2009-04-15 |
JP2010513440A (en) | 2010-04-30 |
EP2121642B1 (en) | 2011-07-27 |
UY30808A1 (en) | 2008-07-31 |
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