AU2003211993A1 - (1,2,4)TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVES - Google Patents

(1,2,4)TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVES

Info

Publication number: AU2003211993A1
Authority: AU; Australia
Prior art keywords: triazolo; pyrimidine derivatives; pyrimidine; derivatives
Prior art date: 2002-02-15
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU2003211993A

Inventor

Hironori Imma

Tomoyuki Kanda

Yoshihisa Kuwana

Junichi Shimada

Shizuo Shiozaki

Tomokazu Watanabe

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

KH Neochem Co Ltd

Original Assignee

Kyowa Hakko Kogyo Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-02-15

Filing date

2003-02-14

Publication date

2003-09-04

2003-02-14 Application filed by Kyowa Hakko Kogyo Co Ltd filed Critical Kyowa Hakko Kogyo Co Ltd

2003-09-04 Publication of AU2003211993A1 publication Critical patent/AU2003211993A1/en

Status Abandoned legal-status Critical Current

Links

QLOWGDIISXJREF-UHFFFAOYSA-N [1,2,4]triazolo[1,5-c]pyrimidine Chemical class C1=CN=CN2N=CN=C21 QLOWGDIISXJREF-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Diabetes (AREA)
Heart & Thoracic Surgery (AREA)
Psychiatry (AREA)
Cardiology (AREA)
Emergency Medicine (AREA)
Obesity (AREA)
Hematology (AREA)
Endocrinology (AREA)
Urology & Nephrology (AREA)
Psychology (AREA)
Hospice & Palliative Care (AREA)
Vascular Medicine (AREA)
Pain & Pain Management (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

AU2003211993A 2002-02-15 2003-02-14 (1,2,4)TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVES Abandoned AU2003211993A1 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
JP2002037819		2002-02-15
JP2002-37819		2002-02-15
PCT/JP2003/001565 WO2003068776A1 (en)	2002-02-15	2003-02-14	[1,2,4]TRIAZOLO[1,5-c]PYRIMIDINE DERIVATIVES

Publications (1)

Publication Number	Publication Date
AU2003211993A1 true AU2003211993A1 (en)	2003-09-04

Family

ID=27678133

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU2003211993A Abandoned AU2003211993A1 (en)	2002-02-15	2003-02-14	(1,2,4)TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVES

Country Status (3)

Country	Link
JP (1)	JPWO2003068776A1 (en)
AU (1)	AU2003211993A1 (en)
WO (1)	WO2003068776A1 (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO2004029056A1 (en) *	2002-09-24	2004-04-08	Kyowa Hakko Kogyo Co., Ltd.	[1,2,4]-TRIAZOLO[1,5-c]PYRIMIDINE DERIVATIVE
WO2004092170A2 (en)	2003-04-09	2004-10-28	Biogen Idec Ma Inc.	Triazolotriazines and pyrazolotriazines useful as a2a adenosine receptor antagon ists
DE602004018637D1 (en) *	2003-04-09	2009-02-05	Biogen Idec Inc	A2A adenosine receptor antagonistic
US7674791B2 (en)	2003-04-09	2010-03-09	Biogen Idec Ma Inc.	Triazolopyrazines and methods of making and using the same
CN101686989B (en)	2007-06-21	2016-10-19	卡拉治疗学股份有限公司	Substituted imidazoheterocycles
US8859538B2 (en)	2007-06-21	2014-10-14	Cara Therapeutics, Inc.	Uses of substituted imidazoheterocycles
SG187502A1 (en)	2008-02-01	2013-02-28	Takeda Pharmaceutical	Oxim derivatives as hsp90 inhibitors
CN107922437B (en) *	2015-09-09	2021-12-10	豪夫迈·罗氏有限公司	Bridged piperidine derivatives
MX2021001186A (en)	2015-11-20	2022-10-11	Forma Therapeutics Inc	Purinones as ubiquitin-specific protease 1 inhibitors.
JP7111733B2 (en)	2017-03-16	2022-08-02	江蘇恒瑞医薬股▲ふん▼有限公司	Heteroaryl[4,3-c]pyrimidin-5-amine derivatives, methods for their preparation, and pharmaceutical uses thereof
US20190292188A1 (en)	2018-02-27	2019-09-26	Incyte Corporation	Imidazopyrimidines and triazolopyrimidines as a2a / a2b inhibitors
US11168089B2 (en)	2018-05-18	2021-11-09	Incyte Corporation	Fused pyrimidine derivatives as A2A / A2B inhibitors
KR20210049090A (en)	2018-07-05	2021-05-04	인사이트 코포레이션	Pyrazine derivatives fused as A2A/A2B inhibitors
EP3883575A4 (en) *	2018-11-20	2022-06-15	Merck Sharp & Dohme Corp.	SUBSTITUTED AMINOTRIAZOLOPYRIMIDINES AND AMINO-TRIAZOLOPYRAZINE ADENOSINE RECEPTOR ANTAGONISTS, PHARMACEUTICAL COMPOSITIONS AND THEIR USE
TWI829857B (en)	2019-01-29	2024-01-21	美商英塞特公司	Pyrazolopyridines and triazolopyridines as a2a / a2b inhibitors
US20240217978A1 (en) *	2021-04-23	2024-07-04	Chong Kun Dang Pharmaceutical Corp.	COMPOUND AS ADENOSINE A2a RECEPTOR ANTAGONIST AND PHARMACEUTICAL COMPOSITION COMPRISING SAME

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ATE257156T1 (en) *	1997-03-24	2004-01-15	Kyowa Hakko Kogyo Kk	(1,2,4)TRIAZOLO(1,5-C)PYRIMIDINE DERIVATIVES
AU756144B2 (en) *	1998-09-22	2003-01-02	Kyowa Hakko Kogyo Co. Ltd.	(1,2,4)triazolo(1,5-c)pyrimidine derivatives

2003
- 2003-02-14 WO PCT/JP2003/001565 patent/WO2003068776A1/en active Application Filing
- 2003-02-14 AU AU2003211993A patent/AU2003211993A1/en not_active Abandoned
- 2003-02-14 JP JP2003567903A patent/JPWO2003068776A1/en not_active Withdrawn

Also Published As

Publication number	Publication date
JPWO2003068776A1 (en)	2005-06-02
WO2003068776A1 (en)	2003-08-21

Legal Events

Date	Code	Title	Description
2004-11-04	MK6	Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase

Publication	Publication Date	Title
AU2003242252A1 (en)	2003-12-22	Bicyclic pyrimidine derivatives
AU2003233519A1 (en)	2003-12-19	Process for imidazo(4,5-c)pyridin-4-amines
EP1599482A4 (en)	2008-10-01	Pyrazolo 1,5-a pyrimidine derivatives
AU2003248588A1 (en)	2004-03-03	Substituted pyrrolopyridines
AU2003292007A1 (en)	2004-06-03	4-AMINO-5-PHENYL-7-CYCLOHEXYL-PYRROLO(2,3-d)PYRIMIDINE DERIVATIVES
EP1416935B8 (en)	2008-08-27	4-amino-6-phenyl-pyrrolo[2,3-d]pyrimidine derivatives
AU2003245700A1 (en)	2003-09-04	Pyrazolopyridine derivatives
AU2003209077A1 (en)	2003-09-02	Pyrimidine compounds
AU2003280680A1 (en)	2004-06-18	Xanthine compound
HK1086012A1 (en)	2006-09-08	8-substitued-6,7,8,9-tetrahydropyrimidoÄ1,2-aÜ pyrimidin-4-one derivatives
HK1088893A1 (en)	2006-11-17	Substituted 8-perfluoroalkyl-6,7,8,9-tetrahydropyrimidoÄ1,2-aÜ pyrimidin-4-one derivatives
AU2003281477A1 (en)	2004-02-09	4-amino-substituted pyrimidine derivatives
AU2003300522A1 (en)	2004-07-22	4-phenyl-pyrimido (4,5-b) indole derivatives
AU2003211993A1 (en)	2003-09-04	(1,2,4)TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVES
AU2003272886A1 (en)	2004-04-19	(1,2,4)-TRIAZOLO(1,5-c)PYRIMIDINE DERIVATIVE
AU2002362806A1 (en)	2003-07-03	Pyrimidine derivatives
AU2003205731A1 (en)	2003-09-04	Mono- and biacylphosphine derivatives
AU2003287992A1 (en)	2004-06-03	Cyclohexylurea derivatives
AU2003208467A1 (en)	2003-09-22	Pyrimidine compounds
AU2003229657A1 (en)	2003-11-10	Triazolopyrimidines
AU2003215676A1 (en)	2003-10-08	Pyrazolopyrimidines derivatives
AU2003222659A1 (en)	2003-11-03	23-o-substituted 5-o-mycaminosyltylonide derivatives
AU2003234131A1 (en)	2003-11-03	5-o-mycaminosyltylonide derivatives
AU2003226725A1 (en)	2003-10-08	Pyrazolopyrimidine derivatives
AU2003223475A1 (en)	2003-11-10	Substituted pyrazine derivatives