+

ZA9810710B - Sustained release formulations comprising alpha-glucosidase-inhibitors - Google Patents

Sustained release formulations comprising alpha-glucosidase-inhibitors

Info

Publication number
ZA9810710B
ZA9810710B ZA9810710A ZA9810710A ZA9810710B ZA 9810710 B ZA9810710 B ZA 9810710B ZA 9810710 A ZA9810710 A ZA 9810710A ZA 9810710 A ZA9810710 A ZA 9810710A ZA 9810710 B ZA9810710 B ZA 9810710B
Authority
ZA
South Africa
Prior art keywords
glucosidase
inhibitors
alpha
sustained release
release formulations
Prior art date
Application number
ZA9810710A
Other languages
English (en)
Inventor
David Goldman
John Amatruda
Carola Portner
Erich Brendel
Patrick Bosche
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of ZA9810710B publication Critical patent/ZA9810710B/xx

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/702Oligosaccharides, i.e. having three to five saccharide radicals attached to each other by glycosidic linkages
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2022Organic macromolecular compounds
    • A61K9/205Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Emergency Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Molecular Biology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
ZA9810710A 1997-11-25 1998-11-24 Sustained release formulations comprising alpha-glucosidase-inhibitors ZA9810710B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US6669897P 1997-11-25 1997-11-25

Publications (1)

Publication Number Publication Date
ZA9810710B true ZA9810710B (en) 1999-06-14

Family

ID=22071124

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA9810710A ZA9810710B (en) 1997-11-25 1998-11-24 Sustained release formulations comprising alpha-glucosidase-inhibitors

Country Status (5)

Country Link
JP (1) JP2001523704A (xx)
AR (1) AR017664A1 (xx)
AU (1) AU1234399A (xx)
WO (1) WO1999026606A2 (xx)
ZA (1) ZA9810710B (xx)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL186223A0 (en) * 2000-05-24 2008-01-20 Pfizer Treatment of rumen acidosis with ??-amylase inhibitors
GB0203296D0 (en) 2002-02-12 2002-03-27 Glaxo Group Ltd Novel composition
US8637512B2 (en) 2002-07-29 2014-01-28 Glaxo Group Limited Formulations and method of treatment
CA2494179C (en) 2002-08-08 2012-04-24 Kissei Pharmaceutical Co., Ltd. Pyrazole derivative, medicinal composition containing the same, medicinal use thereof, and intermediate for production thereof
KR101179451B1 (ko) 2004-03-04 2012-09-07 깃세이 야쿠힌 고교 가부시키가이샤 질소 함유 축합 환 유도체, 그것을 함유하는 의약 조성물및 그 의약 용도
CN102631332A (zh) * 2012-04-28 2012-08-15 邹立兴 一种伏格列波糖片剂及其制备方法
CN104013590A (zh) * 2014-05-09 2014-09-03 万特制药(海南)有限公司 一种含阿卡波糖的药物组合物及其制备方法
WO2016001843A1 (en) * 2014-06-30 2016-01-07 Sun Pharmaceutical Industries Limited Extended-release gastroretentive tablets of voglibose
EA033448B1 (ru) * 2014-12-17 2019-10-31 Empros Pharma Ab Композиция орлистата и акарбозы с модифицированным высвобождением для лечения ожирения и связанных метаболических нарушений
CN110898025A (zh) * 2019-12-12 2020-03-24 湖北欣泽霏药业有限公司 阿卡波糖缓释制剂及其制备方法
CN111265489A (zh) * 2020-03-10 2020-06-12 乐普制药科技有限公司 一种可分割型阿卡波糖微丸缓释片剂

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3134591A1 (de) * 1981-09-01 1983-03-10 Bayer Ag, 5090 Leverkusen Neue arzneimittelpraeparationen fuer glykosidhydrolasen-inhibitoren
EP0194794A3 (en) * 1985-03-08 1986-12-17 Takeda Chemical Industries, Ltd. Saccharide digestion inhibiting composition
DE68905424T2 (de) * 1988-08-22 1993-06-24 Takeda Chemical Industries Ltd Alpha-glucosidaseinhibitor zur foerderung der calciumabsorption.
TW272942B (xx) * 1993-02-10 1996-03-21 Takeda Pharm Industry Co Ltd

Also Published As

Publication number Publication date
WO1999026606A2 (en) 1999-06-03
WO1999026606A3 (en) 1999-08-12
JP2001523704A (ja) 2001-11-27
AU1234399A (en) 1999-06-15
AR017664A1 (es) 2001-09-12

Similar Documents

Publication Publication Date Title
EP1043030A4 (en) MEDICINAL COMPOSITIONS WITH PROLONGED RELEASE
GB9715751D0 (en) Formulations
PL343096A1 (en) Sustained release preparations
IL180864A0 (en) Sustained release ranolazine formulations
EG24198A (en) Extended release formulation
EP1049486A4 (en) GLP-1 FORMULATIONS
SG71879A1 (en) Controlled release compositions
GB9804013D0 (en) Formulations
PL346423A1 (en) Microcapsule formulations
GB2323531B (en) Therapeutic formulations
SG71789A1 (en) Controlled release compositions
HRP20000213B1 (en) Extended release formulation
GB2310860B (en) Stable release agents
PL346414A1 (en) Microcapsule formulations
ZA975703B (en) Sustained release sufentanil compositions
ZA9810710B (en) Sustained release formulations comprising alpha-glucosidase-inhibitors
GB2322867B (en) Release agent
GB9915929D0 (en) Novel release latch-c-i-p
GB9815001D0 (en) Formulations
SI1009387T1 (sl) Stabilizirane tramadolne formulacije s podaljsanim sproscanjem
GB9703099D0 (en) Formulations
GB9703100D0 (en) Formulations
GB9703101D0 (en) Formulations
GB9704521D0 (en) Formulations
GB9816563D0 (en) Controlled release formulations
点击 这是indexloc提供的php浏览器服务,不要输入任何密码和下载