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SV2009003276A - Antagonistas de receptor de orexina de diazepan sustituido - Google Patents

Antagonistas de receptor de orexina de diazepan sustituido

Info

Publication number
SV2009003276A
SV2009003276A SV2009003276A SV2009003276A SV2009003276A SV 2009003276 A SV2009003276 A SV 2009003276A SV 2009003276 A SV2009003276 A SV 2009003276A SV 2009003276 A SV2009003276 A SV 2009003276A SV 2009003276 A SV2009003276 A SV 2009003276A
Authority
SV
El Salvador
Prior art keywords
diazepan
antagonists
replacer
replaced
compounds
Prior art date
Application number
SV2009003276A
Other languages
English (en)
Inventor
Jeffrey M Bergman
Michael J Breslin
Paul J Coleman
Christopher D Cox
Swati P Mercer
Anthony J Roecker
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39284173&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV2009003276(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of SV2009003276A publication Critical patent/SV2009003276A/es

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    • C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
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Abstract

LA PRESENTE INVENCIÓN ESTÁ DIRIGIDA A COMPUESTOS DE DIAZEPAN SUSTITUIDOS QUE SON ANTAGONISTAS DE RECEPTORES DE OREXINA, Y QUE SON ÚTILES EN EL TRATAMIENTO O LA PREVENCIÓN DE TRASTORNOS O ENFERMEDADES NEUROLÓGICOS Y PSIQUIÁTRICOS EN LOS QUE ESTÁN IMPLICADOS LOS RECEPTORES DE OREXINA. LA INVENCIÓN ESTÁ TAMBIÉN DIRIGIDA A COMPOSICIONES FARMACÉUTICAS QUE COMPRENDEN ESTOS COMPUESTOS Y AL USO DE ESTOS COMPUESTOS Y COMPOSICIONES EN LA PREVENCIÓN O EL TRATAMIENTO DE DICHAS ENFERMEDADES EN LAS QUE ESTÁN IMPLICADOS RECEPTORES DE OREXINA
SV2009003276A 2006-12-01 2009-05-27 Antagonistas de receptor de orexina de diazepan sustituido SV2009003276A (es)

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