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EA201300242A1 - Фармацевтические композиции, содержащие замещенные ациланилиды - Google Patents

Фармацевтические композиции, содержащие замещенные ациланилиды

Info

Publication number
EA201300242A1
EA201300242A1 EA201300242A EA201300242A EA201300242A1 EA 201300242 A1 EA201300242 A1 EA 201300242A1 EA 201300242 A EA201300242 A EA 201300242A EA 201300242 A EA201300242 A EA 201300242A EA 201300242 A1 EA201300242 A1 EA 201300242A1
Authority
EA
Eurasian Patent Office
Prior art keywords
pharmaceutical compositions
compositions containing
containing substituted
substituted acylanilides
acylanilides
Prior art date
Application number
EA201300242A
Other languages
English (en)
Other versions
EA024161B1 (ru
Inventor
Джеймс Т. Долтон
Дуэйн Д. Миллер
Original Assignee
Юниверсити Оф Теннесси Рисерч Фаундейшн
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Юниверсити Оф Теннесси Рисерч Фаундейшн filed Critical Юниверсити Оф Теннесси Рисерч Фаундейшн
Publication of EA201300242A1 publication Critical patent/EA201300242A1/ru
Publication of EA024161B1 publication Critical patent/EA024161B1/ru

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/275—Nitriles; Isonitriles
    • A61K31/277—Nitriles; Isonitriles having a ring, e.g. verapamil
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00—Carboxylic acid nitriles
    • C07C255/49—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C255/58—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton
    • C07C255/60—Carboxylic acid nitriles having cyano groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton containing cyano groups and singly-bound nitrogen atoms, not being further bound to other hetero atoms, bound to the carbon skeleton at least one of the singly-bound nitrogen atoms being acylated
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/02—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/32—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C07C235/38—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to acyclic carbon atoms and singly-bound oxygen atoms bound to the same carbon skeleton the carbon skeleton containing six-membered aromatic rings having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
    • A—HUMAN NECESSITIES
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    • A61K31/16—Amides, e.g. hydroxamic acids
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    • A61P3/02—Nutrients, e.g. vitamins, minerals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
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  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Hematology (AREA)
  • Endocrinology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Oncology (AREA)
  • Psychiatry (AREA)
  • Reproductive Health (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Urology & Nephrology (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Communicable Diseases (AREA)
  • Virology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Addiction (AREA)
  • AIDS & HIV (AREA)
  • Emergency Medicine (AREA)
  • Ophthalmology & Optometry (AREA)

Abstract

Изобретение обеспечивает фармацевтические композиции, содержащие замещенные соединения ациланилида, которые применяют для профилактики и/или лечения различных заболеваний или состояний у субъекта, включая рак молочной железы или прогестинзависимые заболевания.
EA201300242A 2006-07-12 2007-07-12 Фармацевтические композиции, содержащие замещенные ациланилиды EA024161B1 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US83015806P 2006-07-12 2006-07-12
US83966506P 2006-08-24 2006-08-24
US90774807P 2007-04-16 2007-04-16

Publications (2)

Publication Number Publication Date
EA201300242A1 true EA201300242A1 (ru) 2013-11-29
EA024161B1 EA024161B1 (ru) 2016-08-31

Family

ID=38923890

Family Applications (3)

Application Number Title Priority Date Filing Date
EA200900177A EA018258B1 (ru) 2006-07-12 2007-07-12 Замещенный ациланилид и содержащие его композиции и способы лечения
EA201690265A EA031888B1 (ru) 2006-07-12 2007-07-12 Способы применения замещенных ациланилидов
EA201300242A EA024161B1 (ru) 2006-07-12 2007-07-12 Фармацевтические композиции, содержащие замещенные ациланилиды

Family Applications Before (2)

Application Number Title Priority Date Filing Date
EA200900177A EA018258B1 (ru) 2006-07-12 2007-07-12 Замещенный ациланилид и содержащие его композиции и способы лечения
EA201690265A EA031888B1 (ru) 2006-07-12 2007-07-12 Способы применения замещенных ациланилидов

Country Status (20)

Country Link
US (1) US20080076828A1 (ru)
EP (2) EP2038252B1 (ru)
JP (5) JP5215300B2 (ru)
KR (2) KR101460693B1 (ru)
CN (1) CN101516840B (ru)
AR (1) AR061980A1 (ru)
AU (1) AU2007272950B2 (ru)
BR (1) BRPI0713179A2 (ru)
CA (1) CA2658394C (ru)
CY (1) CY1118472T1 (ru)
DK (1) DK2038252T3 (ru)
EA (3) EA018258B1 (ru)
ES (2) ES2606313T3 (ru)
HU (1) HUE032274T2 (ru)
IL (3) IL196462A (ru)
LT (1) LT2038252T (ru)
MX (1) MX2009000385A (ru)
PL (1) PL2038252T3 (ru)
PT (1) PT2038252T (ru)
WO (1) WO2008008433A2 (ru)

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