MX9708360A - PYRAZOLO-(1,5a)-PYRIMIDINES, PROCESS FOR PREPARING THE SAME AND THEIR USE. - Google Patents
PYRAZOLO-(1,5a)-PYRIMIDINES, PROCESS FOR PREPARING THE SAME AND THEIR USE.Info
- Publication number
- MX9708360A MX9708360A MX9708360A MX9708360A MX9708360A MX 9708360 A MX9708360 A MX 9708360A MX 9708360 A MX9708360 A MX 9708360A MX 9708360 A MX9708360 A MX 9708360A MX 9708360 A MX9708360 A MX 9708360A
- Authority
- MX
- Mexico
- Prior art keywords
- alkyl
- noch3
- halide
- stands
- hydrogen
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 229910052739 hydrogen Inorganic materials 0.000 abstract 7
- 239000001257 hydrogen Substances 0.000 abstract 7
- 125000003118 aryl group Chemical group 0.000 abstract 6
- -1 cyano, nitro, hydroxy, amino Chemical group 0.000 abstract 6
- 229910052736 halogen Inorganic materials 0.000 abstract 6
- 150000002367 halogens Chemical class 0.000 abstract 6
- 125000001072 heteroaryl group Chemical group 0.000 abstract 6
- 150000002431 hydrogen Chemical class 0.000 abstract 6
- 125000003545 alkoxy group Chemical group 0.000 abstract 5
- 125000000217 alkyl group Chemical group 0.000 abstract 5
- 125000004414 alkyl thio group Chemical group 0.000 abstract 4
- 125000004104 aryloxy group Chemical group 0.000 abstract 4
- 125000005553 heteroaryloxy group Chemical group 0.000 abstract 4
- 125000003342 alkenyl group Chemical group 0.000 abstract 3
- 125000006193 alkinyl group Chemical group 0.000 abstract 3
- 150000001350 alkyl halides Chemical class 0.000 abstract 3
- 125000003710 aryl alkyl group Chemical group 0.000 abstract 3
- 125000005110 aryl thio group Chemical group 0.000 abstract 3
- 125000004093 cyano group Chemical group *C#N 0.000 abstract 3
- 125000004446 heteroarylalkyl group Chemical group 0.000 abstract 3
- 125000005368 heteroarylthio group Chemical group 0.000 abstract 3
- 125000004178 (C1-C4) alkyl group Chemical group 0.000 abstract 2
- 125000002102 aryl alkyloxo group Chemical group 0.000 abstract 2
- 125000000753 cycloalkyl group Chemical group 0.000 abstract 2
- 125000005114 heteroarylalkoxy group Chemical group 0.000 abstract 2
- 125000000623 heterocyclic group Chemical group 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000000547 substituted alkyl group Chemical group 0.000 abstract 2
- WSFSSNUMVMOOMR-UHFFFAOYSA-N Formaldehyde Chemical compound O=C WSFSSNUMVMOOMR-UHFFFAOYSA-N 0.000 abstract 1
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- DBTDEFJAFBUGPP-UHFFFAOYSA-N Methanethial Chemical compound S=C DBTDEFJAFBUGPP-UHFFFAOYSA-N 0.000 abstract 1
- 101100073357 Streptomyces halstedii sch2 gene Proteins 0.000 abstract 1
- 125000003302 alkenyloxy group Chemical group 0.000 abstract 1
- 125000005108 alkenylthio group Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 125000000000 cycloalkoxy group Chemical group 0.000 abstract 1
- 125000005366 cycloalkylthio group Chemical group 0.000 abstract 1
- 125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
- 125000000816 ethylene group Chemical group [H]C([H])([*:1])C([H])([H])[*:2] 0.000 abstract 1
- 125000000219 ethylidene group Chemical group [H]C(=[*])C([H])([H])[H] 0.000 abstract 1
- 235000019256 formaldehyde Nutrition 0.000 abstract 1
- 125000004438 haloalkoxy group Chemical group 0.000 abstract 1
- 125000001188 haloalkyl group Chemical group 0.000 abstract 1
- 125000004995 haloalkylthio group Chemical group 0.000 abstract 1
- 125000005844 heterocyclyloxy group Chemical group 0.000 abstract 1
- 125000004468 heterocyclylthio group Chemical group 0.000 abstract 1
- 125000000956 methoxy group Chemical group [H]C([H])([H])O* 0.000 abstract 1
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 1
- 125000000018 nitroso group Chemical group N(=O)* 0.000 abstract 1
- OSFBJERFMQCEQY-UHFFFAOYSA-N propylidene Chemical compound [CH]CC OSFBJERFMQCEQY-UHFFFAOYSA-N 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Landscapes
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Pyrazolo-(1,5a)-pyrimidines have formula (I), in which the indexes and substituents have the following meanings: n equals 0 or 1; Y stands for 0, S, NRa, OCH2*, SCH2*, NRaCH2*, CH2O*, CH2S*, CH2NRa*, CH2CH2, CRa=Rb or CC, the positions with an * indicating the bond to the phenyl ring; R' stands for H3CO-CO-o=CHOCH3, H3CNH-CO-o=CHOCH3, H3CO-CO-o=NOCH3, H3CNH-CO-o=NOCH3, H2N-CO-o=NOCH3, HO-CO-o=NOCH3, H3CO-CO-o=CHCH3, H3CO-CO-o=CHCH2CH3, H3C-CO-o=CHOCH3, H3C-CO-o=NOCH3, H3CCH2-CO-o=NOCH3, in which o indicates a C atom bound to the phenyl ring, N(OCH3)-CO2CH3, N(CH3)-CO2CH3, N(CH2CH3)-CO2CH3, or a group R'.1-o=NOCH3, R'.2-o=NOCH3, R'.3-o=NOCH3 or R'.4-o=NOCH3; m equals 0, 1, 2 or 3; the residues R" may be different when m is greater than 1; R" stands for cyano, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio or haloalkylthio; R1, R3 stand for hydrogen, cyano, nitro, hydroxy, amino, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkylthio halide, aryl, arylalkyl, aryloxy, arylalkoxy, arylthio, heteroaryl, heteroarylalkyl, heteroaryloxy, heteroarylalkoxy, heteroarylthio or NRcRd, NRcNRdRe, CO-Rc, CO2-Rc, CO-NRcRd, O-CO-Rc, O-CO2-Rc, O-CO-NRcRd, NRc-CO-Rd, NRc-CO2-Rd or NRc-CO-NRdRe; R2 stands for hydrogen, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, aryl, aryloxy, heteroaryl, heteroaryloxy, CO-Rc, CO2-Rc or CRf=NORg; R4 stands for hydrogen, cyano, nitro, nitroso, halogen, alkyl, alkyl halide, alkoxy, alkoxy halide, alkylthio, alkylthio halide, aryl, arylalkyl, aryloxy, arylalkoxy, arylthio, heteroaryl, heteroarylalkyl, heteroaryloxy, heteroarylalkoxy, heteroarylthio or NRcRd, CO-Rc, CO2-Rc or CRf=NORg; Ra, Rb stand for hydrogen, halogen, C1-C4 alkyl or C1-C4 alkyl halide; Rc, Rd and Re stand for hydrogen, alkyl, alkenyl, alkinyl, aryl, arylalkyl, heteroaryl or heteroarylalkyl; Rf stands for hydrogen, cyano, halogen, or optionally substituted alkyl, alkyloxy, alkylthio, alkenyl, alkenyloxy, alkenylthio, alkinyl, alkinyloxy, alkinylthio, cycloalkyl, cycloalkyloxy, cycloalkylthio, heterocyclyl, heterocyclyloxy, heterocyclylthio, aryl, aryloxy, arylthio, heteroaryl, heteroaryloxy or heteroarylthio; Rg stands for hydrogen or optionally substituted alkyl, alkenyl, alkinyl, cycloalkyl, heterocyclyl, aryl or heteroaryl. Also disclosed are a process for preparing the same and their use.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19602072 | 1996-01-20 | ||
| PCT/EP1996/001774 WO1996035690A1 (en) | 1995-05-09 | 1996-04-26 | PYRAZOLO-(1,5a)-PYRIMIDINES, PROCESS FOR PREPARING THE SAME AND THEIR USE |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX9708360A true MX9708360A (en) | 1998-01-31 |
Family
ID=39165744
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX9708360A MX9708360A (en) | 1996-01-20 | 1996-04-26 | PYRAZOLO-(1,5a)-PYRIMIDINES, PROCESS FOR PREPARING THE SAME AND THEIR USE. |
Country Status (1)
| Country | Link |
|---|---|
| MX (1) | MX9708360A (en) |
-
1996
- 1996-04-26 MX MX9708360A patent/MX9708360A/en not_active Application Discontinuation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FA | Abandonment or withdrawal |